SCHEMBL3721044

SCHEMBL3721044

CS(=O)(=O)c1ccc(CN)c(OC(F)(F)F)c1

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.40
SLC6A3 Q01959 1/20 0.40
KCNH2 Q12809 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
CACNA1B Q00975 4/20 0.38
NR1I2 O75469 1/20 0.38
PTGS2 P35354 1/20 0.37
RORC P51449 5/20 0.37
NR1H2 P55055 1/20 0.36
NR1H3 Q13133 1/20 0.36
CYP3A4 P08684 1/20 0.36
HRH4 Q9H3N8 1/20 0.36
PNMT P11086 1/20 0.36
CNR2 P34972 1/20 0.36
BRD4 O60885 1/20 0.35
LRRK2 Q5S007 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14025213 0.81 SMN1; SMN2 (0.54) KCNH2SMN1; SMN2PTGS2
SCHEMBL3713194 0.80 HTR2A (0.35) SLC6A4SLC6A3KCNH2CACNA1BNR1I2
SCHEMBL23143746 0.80 G6PD (0.49) KCNH2TMEM97SIGMAR1SMN1; SMN2CACNA1B
Hydrochloric Acid SCHEMBL4916424 0.80 SMN1; SMN2 (0.53) KCNH2SMN1; SMN2PTGS2
SCHEMBL18230961 0.78 FFAR4 (0.43) KCNH2TMEM97SIGMAR1SMN1; SMN2CACNA1B
SCHEMBL3710331 0.76 KIF11 (0.46) KCNH2PTGS2NR1H2NR1H3HRH4
SCHEMBL18230946 0.76 MAPT (0.44) SLC6A4SLC6A3KCNH2TMEM97SIGMAR1
SCHEMBL24254583 0.76 SMN1; SMN2 (0.45) SLC6A4SLC6A3KCNH2TMEM97SIGMAR1
SCHEMBL23155765 0.74 LRRK2 (0.46) KCNH2TMEM97SIGMAR1SMN1; SMN2PTGS2
SCHEMBL3711714 0.74 IDO1 (0.42) SLC6A4SLC6A3KCNH2HRH4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO claimed
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed