SCHEMBL3721096

SCHEMBL3721096

CC(Nc1nc(CN)cc(-c2ccc(C(F)(F)F)cc2)n1)c1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
IDH1 O75874 4/20 0.46
MAPK13 O15264 3/20 0.44
MAPK12 P53778 3/20 0.44
MAPK11 Q15759 3/20 0.44
MAPK14 Q16539 3/20 0.44
KCNH3 Q9ULD8 1/20 0.43
CASR P41180 4/20 0.41
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
ATP1A1 P05023 1/20 0.40
ATP1B1 P05026 1/20 0.40
ATP1A3 P13637 1/20 0.40
ATP1B2 P14415 1/20 0.40
ATP1A2 P50993 1/20 0.40
ATP1B3 P54709 1/20 0.40
FXYD2 P54710 1/20 0.40
ATP1A4 Q13733 1/20 0.40
FAAH O00519 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3723210 0.85 ADORA2B (0.41)
SCHEMBL3724702 0.81 CTSS (0.47)
SCHEMBL3721092 0.81 SCN9A (0.50) IDH1MAPK14KCNH3
SCHEMBL3722102 0.80 TRPV3 (0.53)
SCHEMBL3727421 0.78 CTSS (0.41) FAAH
SCHEMBL3721028 0.78 ADORA1 (0.48) MAPK14
SCHEMBL7028475 0.74 LCK (0.59) MAPK13MAPK12MAPK11MAPK14ATP1A1
SCHEMBL3717583 0.74 PTGS1 (0.56)
SCHEMBL3725441 0.74 IDH2 (0.48) IDH1
SCHEMBL3725421 0.73 DPP4 (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed