SCHEMBL3722079

SCHEMBL3722079

COc1ccc(Oc2cnc(N(C)C(=O)C3(NC(=O)c4cc(OC)no4)CC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.37

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 14/20 0.37
BDKRB1 P46663 3/20 0.36
GAA P10253 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721992 0.93 BDKRB1 (0.35) CNR1BDKRB1GAA
SCHEMBL3728529 0.89 MEN1 (0.43) BDKRB1GAA
SCHEMBL3722724 0.86 MEN1 (0.36) CNR1BDKRB1GAA
SCHEMBL3722078 0.84 BDKRB1 (0.40) CNR1BDKRB1
SCHEMBL3725869 0.82 MEN1 (0.42) BDKRB1
SCHEMBL765813 0.81 CNR1 (0.42) CNR1BDKRB1
Trifluoroacetic Acid SCHEMBL3718216 0.81 CNR1 (0.47) CNR1BDKRB1
SCHEMBL3722860 0.80 GAA (0.33) GAA
SCHEMBL3721990 0.79 BDKRB1 (0.37) CNR1BDKRB1
SCHEMBL3719005 0.77 MAPK10 (0.35) GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed