SCHEMBL3721992

SCHEMBL3721992

COc1ccc(Oc2cnc(N(C)C(=O)C3(NC(=O)c4cc(OC)no4)CCOC3)nc2)c(C(F)(F)F)c1

nearest known ligand 0.35

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
BDKRB1 P46663 8/20 0.35
CNR1 P21554 7/20 0.33
GAA P10253 1/20 0.33
TP53 P04637 1/20 0.32
MAPK8 P45983 1/20 0.32
MAPK10 P53779 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3722079 0.93 CNR1 (0.37) BDKRB1CNR1GAA
SCHEMBL3725869 0.90 MEN1 (0.42) BDKRB1TP53MAPK8MAPK10
SCHEMBL3721990 0.86 BDKRB1 (0.37) BDKRB1CNR1TP53
SCHEMBL3725887 0.82 MAPK10 (0.31) GAAMAPK8MAPK10
SCHEMBL3728529 0.82 MEN1 (0.43) BDKRB1GAAMAPK8MAPK10
SCHEMBL3722724 0.79 MEN1 (0.36) BDKRB1CNR1GAATP53MAPK8
SCHEMBL3722078 0.79 BDKRB1 (0.40) BDKRB1CNR1
Trifluoroacetic Acid SCHEMBL3718216 0.76 CNR1 (0.47) BDKRB1CNR1
SCHEMBL765813 0.76 CNR1 (0.42) BDKRB1CNR1
SCHEMBL3725868 0.75 MEN1 (0.41) BDKRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed