SCHEMBL3722137

SCHEMBL3722137

COC(=O)c1ccc(-c2cc(C#N)c(C#N)cc2-c2ccc(C(=O)OC)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.51
CA1 P00915 4/20 0.47
CA2 P00918 4/20 0.47
CA12 O43570 3/20 0.47
CA9 Q16790 3/20 0.47
CA14 Q9ULX7 3/20 0.47
CA7 P43166 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
PTGS2 P35354 1/20 0.46
PTGS1 P23219 1/20 0.44
ERN1 O75460 1/20 0.44
TSHR P16473 1/20 0.44
TBK1 Q9UHD2 1/20 0.44
SLC2A1 P11166 1/20 0.44
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
XDH P47989 1/20 0.43
KDM4E B2RXH2 1/20 0.43
SETD7 Q8WTS6 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28577777 0.87 EGFR (0.52) EGFRCA1CA2CA12CA9
SCHEMBL3717515 0.85 ERN1 (0.50) EGFRCA1CA2CA12CA9
SCHEMBL6165708 0.84 ESR2 (0.56) EGFRCA1CA2CA12CA9
SCHEMBL21261147 0.84 EGFR (0.62) EGFRCA1CA2CA12CA9
SCHEMBL9041238 0.83 EGFR (0.44) EGFRCA1CA2CA12CA9
SCHEMBL15999096 0.82 PTGS1 (0.51) EGFRPTGS1ERN1SLC2A1MAPT
SCHEMBL21083536 0.81 EGFR (0.64) EGFRPTGS2ERN1TSHRSLC2A1
SCHEMBL30849990 0.81 EGFR (0.64) EGFRPTGS2ERN1TSHRSLC2A1
SCHEMBL8148281 0.81 CA1 (0.52) CA1CA2CA12CA9CA14
SCHEMBL28577779 0.80 EGFR (0.49) EGFRPTGS2XDHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010136178-A1 THE PREPARATION OF A DYE COMPOUND AND A METHOD FOR MAKING THE SAME CORUS UK LIMITED (GB) 2010-12-02 WO disclosed