SCHEMBL28577779

SCHEMBL28577779

COC(=O)c1ccc(-c2ccc(C(=O)O)cc2)c(C#N)c1

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.49
PTGS2 P35354 1/20 0.47
GRM5 P41594 1/20 0.46
XDH P47989 3/20 0.45
CYP2C8 P10632 1/20 0.44
PRKAB2 O43741 1/20 0.43
PRKAG1 P54619 1/20 0.43
PRKAA2 P54646 1/20 0.43
PRKAA1 Q13131 1/20 0.43
PRKAG3 Q9UGI9 1/20 0.43
PRKAG2 Q9UGJ0 1/20 0.43
PRKAB1 Q9Y478 1/20 0.43
KDM4E B2RXH2 1/20 0.42
KDM6B O15054 1/20 0.42
KDM5C P41229 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
KDM2A Q9Y2K7 1/20 0.42
KDM3A Q9Y4C1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28577777 0.93 EGFR (0.52) EGFRPTGS2GRM5XDHKDM4E
SCHEMBL404224 0.90 EGFR (0.57) EGFRPTGS2GRM5XDH
SCHEMBL28571512 0.86 XDH (0.48) GRM5XDH
SCHEMBL28880690 0.86 CA1 (0.50) EGFRXDHKDM4E
SCHEMBL23768092 0.84 XDH (0.51) EGFRXDHCYP2C8
SCHEMBL29788308 0.83 CYP2C8 (0.56) XDHCYP2C8PRKAB2PRKAG1PRKAA2
SCHEMBL2041742 0.83 CYP2C8 (0.56) XDHCYP2C8PRKAB2PRKAG1PRKAA2
SCHEMBL15999096 0.82 PTGS1 (0.51) EGFRGRM5KDM4E
SCHEMBL8176629 0.81 GRM5 (0.49) GRM5XDHKDM4E
SCHEMBL3722137 0.80 EGFR (0.51) EGFRPTGS2XDHKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113024382-A Monocyano-substituted polycarboxylic organic ligand and preparation method thereof 同济大学 2021-06-25 CN disclosed