SCHEMBL3723398

SCHEMBL3723398

CC(C(=O)O)c1cncc(-c2ccc(C(F)(F)F)cc2)c1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 11/20 0.56
AKR1C2 P52895 11/20 0.56
PTGS2 P35354 3/20 0.53
PSEN1 P49768 1/20 0.53
PSEN2 P49810 1/20 0.53
APH1B Q8WW43 1/20 0.53
NCSTN Q92542 1/20 0.53
APH1A Q96BI3 1/20 0.53
PSENEN Q9NZ42 1/20 0.53
MMP1 P03956 1/20 0.43
MMP2 P08253 1/20 0.43
MMP3 P08254 1/20 0.43
MMP7 P09237 1/20 0.43
MMP9 P14780 1/20 0.43
MMP13 P45452 1/20 0.43
KDM1A O60341 1/20 0.43
HDAC1 Q13547 1/20 0.43
MAP4K4 O95819 1/20 0.42
FFAR1 O14842 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29010056 0.82 AKR1C3 (0.47) AKR1C3AKR1C2PTGS2
SCHEMBL6270587 0.80 AKR1C3 (0.63) AKR1C3AKR1C2PTGS2PSEN1PSEN2
SCHEMBL11960749 0.78 AKR1C3 (0.60) AKR1C3AKR1C2PTGS2PSEN1PSEN2
SCHEMBL1797371 0.77 AKR1C3 (0.65) AKR1C3AKR1C2PTGS2PSEN1PSEN2
SCHEMBL31301420 0.75 MKNK1 (0.62) KDM1AHDAC1MAP4K4
SCHEMBL1843427 0.75 MKNK1 (0.62) KDM1AHDAC1MAP4K4
SCHEMBL2161512 0.74 AKR1C3 (0.59) AKR1C3AKR1C2PTGS2PSEN1PSEN2
SCHEMBL13876033 0.72 KDM1A (0.54) KDM1AHDAC1MAP4K4
SCHEMBL1372793 0.72 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2PSEN1PSEN2
SCHEMBL9895027 0.71 RXRA (0.57) PSEN1PSEN2APH1BNCSTNAPH1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2435428-B1 SUBSTITUTED PIPERIDINES BAYER IP GMBH (DE) 2013-07-31 EP disclosed
WO-2010136128-A1 SUBSTITUTED PIPERIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-12-02 WO disclosed