SCHEMBL3725438

SCHEMBL3725438

CC(C)(O)CNc1nc(C(N)=O)cc(-c2ccc(C(F)(F)F)cc2)n1

nearest known ligand 0.47

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 14/20 0.47
IDH2 P48735 2/20 0.47
FPR2 P25090 4/20 0.45
ADORA3 P0DMS8 1/20 0.44
VCP P55072 1/20 0.43
CASP1 P29466 1/20 0.42
IDH1 O75874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724700 0.85 SCN9A (0.51) SCN9AFPR2ADORA3CASP1
SCHEMBL3727419 0.85 SCN9A (0.52) SCN9AFPR2ADORA3VCPCASP1
SCHEMBL3717581 0.84 PTGS1 (0.56) SCN9AFPR2ADORA3VCPCASP1
SCHEMBL3725441 0.82 IDH2 (0.48) IDH2ADORA3VCPIDH1
SCHEMBL3721124 0.80 MAPT (0.64)
SCHEMBL3718623 0.78 KDM4E (0.58) SCN9AVCP
SCHEMBL3717789 0.78 SCN9A (0.53) SCN9A
SCHEMBL3722100 0.78 SCN9A (0.52) SCN9AFPR2
SCHEMBL3727125 0.78 PTGS2 (0.48) SCN9AFPR2ADORA3VCPCASP1
SCHEMBL3720230 0.78 VCP (0.51) SCN9AFPR2VCP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US claimed
US-8614201-B2 Heterocyclic amides as modulators of TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2013-12-24 US disclosed
WO-2010141805-A1 HETEROCYCLIC AMIDES AS MODULATORS OF TRPA1 JANSSEN PHARMACEUTICA NV (BE) 2010-12-09 WO disclosed