SCHEMBL3725903

SCHEMBL3725903

COc1ccc(Oc2cnc(C#N)c(Cl)c2)c(C(F)(F)F)c1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SLC22A12 Q96S37 2/20 0.45
AR P10275 14/20 0.44
MAPK8 P45983 1/20 0.40
MAPK10 P53779 1/20 0.40
CTSS P25774 2/20 0.39
CTSK P43235 2/20 0.39
PGR P06401 1/20 0.39
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
OPRK1 P41145 1/20 0.38
HTT P42858 1/20 0.38
RAB9A P51151 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719152 0.82 AR (0.48) SLC22A12ARCTSSCTSKPGR
SCHEMBL3730195 0.82 AR (0.48) SLC22A12ARCTSSPGR
SCHEMBL3722067 0.79 MAPK10 (0.42) MAPK8MAPK10MAPTRAB9A
SCHEMBL672513 0.77 SRC (0.40) ARMAPK8MAPK10PGRNPC1
SCHEMBL1006358 0.76 MAPT (0.46) SLC22A12NPC1ALDH1A1LMNAMAPT
SCHEMBL756605 0.76 AR (0.52) ARPGRRAB9A
SCHEMBL3725849 0.76 AR (0.44) ARMAPK8MAPK10CTSSPGR
SCHEMBL24424820 0.75 AR (0.44) ARCTSSCTSKPGRMAPT
Trifluoroacetic Acid SCHEMBL3720595 0.73 MAPK10 (0.44) MAPK8MAPK10LMNA
SCHEMBL15096357 0.73 AR (0.60) ARPGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed