SCHEMBL3730195

SCHEMBL3730195

COc1ccc(Oc2ccc(C#N)nc2)c(C(F)(F)F)c1

nearest known ligand 0.48

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AR P10275 15/20 0.48
PGR P06401 2/20 0.43
CTSS P25774 1/20 0.43
SLC22A12 Q96S37 2/20 0.42
NQO1 P15559 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3719152 0.87 AR (0.48) ARPGRCTSSSLC22A12
SCHEMBL3725849 0.86 AR (0.44) ARPGRCTSS
SCHEMBL3725903 0.82 SLC22A12 (0.45) ARPGRCTSSSLC22A12
SCHEMBL756605 0.81 AR (0.52) ARPGR
SCHEMBL3723563 0.81 NQO1 (0.44) ARSLC22A12NQO1
SCHEMBL3726572 0.79 NQO1 (0.43) ARSLC22A12NQO1
SCHEMBL3722579 0.78 L3MBTL1 (0.40) AR
SCHEMBL3726016 0.78 L3MBTL1 (0.40) AR
SCHEMBL3718921 0.78 L3MBTL1 (0.40) AR
SCHEMBL3727500 0.77 MAPK10 (0.40)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010097373-A1 COMPOUNDS FOR USE AS BRADYKININ B1 ANTAGONISTS BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2010-09-02 WO disclosed