SCHEMBL3726481

SCHEMBL3726481

O=C(Cl)c1cccc([N+](=O)[O-])c1-c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FBP1 P09467 1/20 0.49
TSHR P16473 1/20 0.49
CTSD P07339 1/20 0.49
ALDH1A1 P00352 3/20 0.47
TDP1 Q9NUW8 2/20 0.47
CRHBP P24387 1/20 0.44
CRHR2 Q13324 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.43
GPR35 Q9HC97 1/20 0.43
TP53 P04637 1/20 0.43
S100A4 P26447 2/20 0.42
PTPRC P08575 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL593074 0.87 TSHR (0.60) FBP1TSHRCTSDALDH1A1TDP1
SCHEMBL299878 0.84 FBP1 (0.49) FBP1TSHRCTSDALDH1A1TDP1
SCHEMBL28149001 0.83 CTSD (0.69) FBP1TSHRCTSDALDH1A1TDP1
SCHEMBL10477073 0.81 ALDH1A1 (0.53) FBP1TSHRCTSDALDH1A1TDP1
SCHEMBL103644 0.81 CTSD (0.65) TSHRCTSDALDH1A1TDP1CYP1A2
SCHEMBL28221727 0.80 TDP1 (0.63) FBP1TSHRALDH1A1TDP1CRHBP
SCHEMBL10718417 0.80 ALDH1A1 (0.50) TSHRALDH1A1TDP1KDM4EMAPT
SCHEMBL16719902 0.80 TSHR (0.53) FBP1TSHRCTSDALDH1A1TDP1
SCHEMBL16120074 0.80 SLC6A2 (0.58) FBP1TSHRCTSDALDH1A1TDP1
Hydrochloric Acid SCHEMBL10567555 0.79 CTSD (0.62) TSHRCTSDALDH1A1TDP1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010120987-A1 RING FUSED, UREIDOARYL- AND CARBAMOYLARYL-BRIDGED MORPHOLINO-PYRIMIDINE COMPOUNDS, THEIR USE AS MTOR KINASE AND PI3 KINASE INHIBITORS, AND THEIR SYNTHESES WYETH LLC (US) 2010-10-21 WO disclosed