SCHEMBL3726792

SCHEMBL3726792

CC(=O)c1ccc2nc(Oc3ccc(OCCN(C)C)cc3C)ccc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.45
KDM4E B2RXH2 4/20 0.44
ALDH1A1 P00352 4/20 0.44
THRA P10827 3/20 0.41
TDP1 Q9NUW8 1/20 0.40
DRD3 P35462 3/20 0.40
ADRA2A P08913 2/20 0.40
ADRA2B P18089 2/20 0.40
ADRA2C P18825 2/20 0.40
HTR2C P28335 2/20 0.40
HRH1 P35367 2/20 0.40
MCHR1 Q99705 2/20 0.40
CHRM2 P08172 1/20 0.40
CHRM1 P11229 1/20 0.40
DRD1 P21728 1/20 0.40
HRH2 P25021 1/20 0.40
HTR1B P28222 1/20 0.40
HTR2A P28223 1/20 0.40
MCHR2 Q969V1 1/20 0.40
THRB P10828 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3724671 0.95 PDE4B (0.44) PDE4BKDM4EALDH1A1THRATHRB
SCHEMBL3720755 0.90 PDE4B (0.46) PDE4BALDH1A1THRAMEN1KMT2A
SCHEMBL3724295 0.84 PDE4B (0.46) PDE4BALDH1A1MCHR1THRBGAA
SCHEMBL3724232 0.83 PDE4B (0.46) PDE4BALDH1A1MCHR1GAAMAPT
SCHEMBL3718228 0.82 ACACB (0.42) KDM4EALDH1A1DRD3ADRA2AADRA2B
SCHEMBL3718230 0.82 MTNR1A (0.48) KDM4EALDH1A1DRD3DRD2HRH3
SCHEMBL3721868 0.82 PDE4B (0.48) PDE4BALDH1A1MEN1KMT2AMAPT
SCHEMBL3726793 0.82 ADRB2 (0.40) KDM4EALDH1A1TDP1DRD3DRD2
SCHEMBL3721926 0.81 PDE4B (0.44) PDE4BMCHR1
SCHEMBL3719225 0.80 PDE4B (0.46) PDE4BALDH1A1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed