SCHEMBL3724232

SCHEMBL3724232

CC(=O)c1ccc2nc(Oc3ccc(OCC4CC4)cc3C)ccc2c1

nearest known ligand 0.46

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PDE4B Q07343 1/20 0.46
ACACB O00763 6/20 0.45
CYP3A4 P08684 2/20 0.41
ACACA Q13085 2/20 0.41
CYP2C9 P11712 1/20 0.41
PARP15 Q460N3 1/20 0.39
PARP10 Q53GL7 1/20 0.39
PARP2 Q9UGN5 1/20 0.39
KDM2B Q8NHM5 1/20 0.39
MCHR1 Q99705 8/20 0.39
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
PPARG P37231 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721926 0.95 PDE4B (0.44) PDE4BACACBCYP3A4ACACACYP2C9
SCHEMBL3720427 0.89 ACACB (0.56) PDE4BACACBCYP3A4ACACACYP2C9
SCHEMBL3719578 0.87 PDE4B (0.53) PDE4BACACBACACAPARP15PARP10
SCHEMBL3721101 0.85 PDE4B (0.44) PDE4BACACBCYP3A4ACACACYP2C9
SCHEMBL3720755 0.85 PDE4B (0.46) PDE4BALDH1A1GAAMAPTL3MBTL1
SCHEMBL3797155 0.84 MTNR1A (0.42) PDE4BACACBCYP3A4ACACACYP2C9
SCHEMBL3724295 0.84 PDE4B (0.46) PDE4BACACBMCHR1ALDH1A1GAA
SCHEMBL3727011 0.83 PDE4B (0.50) PDE4BACACBPARP15PARP10PARP2
SCHEMBL3725384 0.83 PDE4B (0.50) PDE4BACACBCYP3A4ACACACYP2C9
SCHEMBL3726792 0.83 PDE4B (0.45) PDE4BMCHR1ALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed