SCHEMBL3727697

SCHEMBL3727697

CC(C)Sc1ccc(Oc2ccc3cc(CCN)ccc3n2)c(Br)c1

nearest known ligand 0.34

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
TSHR P16473 1/20 0.34
NFKB1 P19838 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ATM Q13315 1/20 0.33
MEN1 O00255 1/20 0.33
LMNA P02545 1/20 0.33
APEX1 P27695 1/20 0.33
KMT2A Q03164 1/20 0.33
GLA P06280 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3720189 0.88 TSHR (0.34) CYP1A2CYP3A4TSHRNFKB1KDM4E
SCHEMBL3720478 0.88 GLA (0.40) CYP1A2CYP3A4TSHRNFKB1KDM4E
SCHEMBL3720538 0.85 LMNA (0.31) CYP1A2LMNASMN1; SMN2
SCHEMBL3716750 0.84 CYP1A2 (0.35) CYP1A2CYP3A4TSHRNFKB1MEN1
SCHEMBL3718486 0.82 TSHR (0.37) CYP1A2CYP3A4TSHRNFKB1KDM4E
SCHEMBL3722863 0.81 CYP1A2 (0.34) CYP1A2CYP3A4TSHRNFKB1KDM4E
SCHEMBL3727138 0.80 TSHR (0.34) CYP1A2CYP3A4TSHRNFKB1KDM4E
SCHEMBL3727694 0.79 MAPT (0.32) CYP1A2LMNASMN1; SMN2
SCHEMBL3717625 0.79 S1PR3 (0.36) CYP1A2CYP3A4TSHRNFKB1KDM4E
SCHEMBL3717501 0.79 GLA (0.39) CYP1A2CYP3A4TSHRNFKB1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010127208-A1 INHIBITORS OF ACETYL-COA CARBOXYLASE FOREST LABORATORIES HOLDINGS LIMITED (BM) 2010-11-04 WO disclosed