SCHEMBL3728686

SCHEMBL3728686

Cc1nc2ccccc2n1-c1ccc(NC2CCN(C(=O)OC(C)(C)C)CC2)cc1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.57
MAPT P10636 2/20 0.56
MAPK1 P28482 2/20 0.56
NPC1 O15118 1/20 0.56
HTT P42858 1/20 0.56
RAB9A P51151 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.56
CNR1 P21554 1/20 0.49
CNR2 P34972 1/20 0.49
HRH3 Q9Y5N1 4/20 0.49
GPR119 Q8TDV5 5/20 0.47
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
OGFRL1 Q5TC84 1/20 0.47
BRD4 O60885 1/20 0.45
KDM4E B2RXH2 1/20 0.44
HPGD P15428 1/20 0.44
TSHR P16473 1/20 0.44
ATM Q13315 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3805262 0.94 HRH3 (0.50) ALDH1A1MAPTMAPK1NPC1HTT
SCHEMBL3805265 0.94 HRH3 (0.50) ALDH1A1MAPTMAPK1NPC1HTT
SCHEMBL3728687 0.87 HRH3 (0.64) MAPTHRH3GPR119KDM4E
SCHEMBL3724630 0.84 MMP7 (0.57) ALDH1A1MAPTMAPK1NPC1HTT
SCHEMBL3639498 0.83 HRH3 (0.67) HRH3
SCHEMBL3668354 0.83 HRH3 (0.67) HRH3
SCHEMBL3639495 0.83 HRH3 (0.67) HRH3
SCHEMBL16149777 0.83 HRH3 (0.57) ALDH1A1MAPK1HTTCNR2HRH3
SCHEMBL3726061 0.80 ALDH1A1 (0.45) ALDH1A1MAPTMAPK1NPC1HTT
SCHEMBL3726059 0.80 ALDH1A1 (0.45) ALDH1A1MAPTMAPK1NPC1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2155719-A1 AZACYCLYLBENZAMIDE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS Wyeth LLC (US) 2010-02-24 EP disclosed
WO-2008147945-A1 AZACYCLYLBENZAMIDE DERIVATIVES AS HISTAMINE-3 ANTAGONISTS WYETH (US) 2008-12-04 WO disclosed