SCHEMBL3728799

SCHEMBL3728799

O=C(O)CCc1ccccc1CO

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4F2 P78329 2/20 0.58
CYP4A11 Q02928 2/20 0.58
KEAP1 Q14145 1/20 0.56
FFAR1 O14842 8/20 0.53
PTGER1 P34995 3/20 0.51
PTGER4 P35408 3/20 0.51
PTGER3 P43115 3/20 0.51
PTGER2 P43116 3/20 0.51
PARP1 P09874 1/20 0.49
HDAC3 O15379 1/20 0.47
MAPK1 P28482 1/20 0.47
ADRA1A P35348 1/20 0.47
HDAC4 P56524 1/20 0.47
SLC6A3 Q01959 1/20 0.47
HDAC1 Q13547 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
HDAC7 Q8WUI4 1/20 0.47
HDAC2 Q92769 1/20 0.47
HDAC10 Q969S8 1/20 0.47
HDAC11 Q96DB2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9566135 0.94 CYP4F2 (0.53) CYP4F2CYP4A11KEAP1FFAR1PTGER1
SCHEMBL59198 0.91 KEAP1 (0.65) KEAP1FFAR1PTGER1PTGER4PTGER3
SCHEMBL8573204 0.87 KEAP1 (0.56) CYP4F2CYP4A11KEAP1FFAR1PTGER1
SCHEMBL10704357 0.84 MAPT (0.61) CYP4F2CYP4A11HDAC3MAPK1ADRA1A
SCHEMBL11719124 0.84 MAPT (0.61) CYP4F2CYP4A11HDAC3MAPK1ADRA1A
SCHEMBL9566173 0.83 HDAC3 (0.53) CYP4F2CYP4A11KEAP1FFAR1HDAC3
SCHEMBL29373796 0.83 AKR1B1 (0.65) KEAP1FFAR1PTGER1PTGER4PTGER3
SCHEMBL35529 0.83 AKR1B1 (0.65) KEAP1FFAR1PTGER1PTGER4PTGER3
SCHEMBL878984 0.83 KEAP1 (0.56) CYP4F2CYP4A11KEAP1FFAR1PTGER1
SCHEMBL7128255 0.83 AKR1B1 (0.65) KEAP1FFAR1PTGER1PTGER4PTGER3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2238107-A1 PROCESS FOR THE MANUFACTURE OF A 6-FLUORO-1,2-DIHYDRO-2-OXO-3H-INDOL-3-YLIDENE DERIVATIVE Boehringer Ingelheim International GmbH (DE) 2010-10-13 EP claimed
WO-2009092580-A1 PROCESS FOR THE MANUFACTURE OF A 6-FLUORO-1,2-DIHYDRO-2-OXO-3H-INDOL-3-YLIDENE DERIVATIVE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-07-30 WO claimed
US-4731126-A HYDROXYMETHYL CARBOXYLIC ACID THE DOW CHEMICAL COMPANY (US) 1988-03-15 US claimed
US-11746364-B2 Enzymatic synthesis of kavalactones and flavokavains WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2023-09-05 US disclosed
US-11739354-B2 Enzymatic synthesis of kavalactones and flavokavains WHITEHEAD INSTITUTE FOR BIOMEDICAL RESEARCH (US) 2023-08-29 US disclosed
WO-2008009735-A1 PYRAZOLO (3, 4-B) PYRIDINE DERIVATIVES AS PDE4 INHIBITORS GLAXO GROUP LIMITED (GB) 2008-01-24 WO disclosed
CN-1931821-A Process of resolving optical isomer of 2-hydroxmethyl-3-phenylpropionic acid SHANGHAI INST OF MEDICINE INDU (CN) 2007-03-21 CN disclosed
US-5280034-A Bis-heterocyclic prostaglandin analogs E. R. SQUIBB & SONS, INC. (US) 1994-01-18 US disclosed
US-4731126-A HYDROXYMETHYL CARBOXYLIC ACID THE DOW CHEMICAL COMPANY (US) 1988-03-15 US disclosed