Chlormadinone

Chlormadinone

SCHEMBL37291

CC(=O)[C@@]1(O)CC[C@H]2[C@@H]3C=C(Cl)C4=CC(=O)CC[C@]4(C)[C@H]3CC[C@@]21C

nearest known ligand 0.78

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 4/20 0.78
AR P10275 3/20 0.78
CHRM1 P11229 2/20 0.78
NR3C1 P04150 5/20 0.71
SMN1; SMN2 Q16637 5/20 0.71
CYP3A4 P08684 5/20 0.71
HIF1A Q16665 5/20 0.71
CYP2C19 P33261 3/20 0.71
ADORA3 P0DMS8 2/20 0.71
MAPK1 P28482 2/20 0.71
NPSR1 Q6W5P4 2/20 0.71
ALDH1A1 P00352 2/20 0.71
CHRM2 P08172 1/20 0.71
THRB P10828 1/20 0.71
TBXA2R P21731 1/20 0.71
ADRA1A P35348 1/20 0.71
USP2 O75604 1/20 0.71
DRD1 P21728 1/20 0.63
OPRK1 P41145 1/20 0.63
PDE3A Q14432 1/20 0.63

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Chlormadinone SCHEMBL13358512 1.00 PGR (0.78) PGRARCHRM1NR3C1SMN1; SMN2
SCHEMBL8942 0.88 PGR (1.00) PGRARCHRM1NR3C1SMN1; SMN2
SCHEMBL2294866 0.88 PGR (1.00) PGRARCHRM1NR3C1SMN1; SMN2
SCHEMBL16690685 0.88 PGR (1.00) PGRARCHRM1NR3C1SMN1; SMN2
SCHEMBL5020044 0.88 PGR (1.00) PGRARCHRM1NR3C1SMN1; SMN2
SCHEMBL11510962 0.87 PGR (0.78) PGRARCHRM1NR3C1SMN1; SMN2
SCHEMBL11407502 0.86 PGR (0.65) PGRARCHRM1NR3C1SMN1; SMN2
Acetic Acid SCHEMBL25192781 0.86 PGR (0.96) PGRARCHRM1NR3C1SMN1; SMN2
SCHEMBL8623116 0.85 PGR (0.75) PGRARCHRM1NR3C1SMN1; SMN2
Acetic Acid SCHEMBL28104035 0.85 PGR (0.94) PGRARCHRM1NR3C1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 4054 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4440706-B1 COMPOSITIONS FOR PROMOTING HAIR GROWTH ESTETRA SRL (BE) 2026-04-29 EP claimed
EP-4525938-B1 RADIOPHARMACEUTICAL COMPLEXES TARGETING PROSTATE-SPECIFIC MEMBRANE ANTIGEN AND ITS COMBINATIONS BAYER AG (DE) 2026-03-11 EP claimed
EP-4463570-B1 METHOD FOR HORMONE OR DRUG SCREENING IN A TISSUE SAMPLE ECOLE POLYTECHNIQUE FED LAUSANNE EPFL (CH) 2026-01-14 EP claimed
EP-4637777-A1 USE OF ESTETROL IN HEPATICALLY IMPAIRED PATIENTS Estetra SRL (BE) 2025-10-29 EP claimed
US-20250295634-A1 USE OF ANTIANDROGENS TO TREAT SEPSIS RHODE ISLAND HOSPITAL 2025-09-25 US claimed
EP-4602049-A1 SOS1 INHIBITORS Bayer Aktiengesellschaft (DE) 2025-08-20 EP claimed
US-20250255968-A1 INTRAVAGINAL DEVICES FOR DRUG DELIVERY KISER PATRICK F (US) 2025-08-14 US claimed
EP-4587439-A1 SULFONE-SUBSTITUTED PYRIDO[3,4-D]PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF CANCER Bayer Aktiengesellschaft (DE) 2025-07-23 EP claimed
US-20250195450-A1 BIOERODIBLE DRUG DELIVERY IMPLANTS HERA HEALTH SOLUTIONS INC. 2025-06-19 US claimed
US-12318395-B2 Ethinyl estradiol-β-cyclodextrin complex and process for preparing thereof LABORATORIOS LEON FARMA, S.A. (ES) 2025-06-03 US claimed
WO-1992015289-A1 COMPOSITIONS AND METHODS FOR TOPICAL ADMINISTRATION OF PHARMACEUTICALLY ACTIVE AGENTS NOVEN PHARMACEUTICALS, INC. (US) 1992-09-17 WO claimed
EP-0491803-A1 IMPLANTABLE DELIVERY DISPENSER. ALZA CORP (US) 1992-07-01 EP claimed
US-5112614-A IMPLANTABLE DELIVERY DISPENSER ALZA CORPORATION (US) 1992-05-12 US claimed
EP-0198893-B1 HAIR GROWTH MODIFICATION HANDELMAN, Joseph H. (US) 1992-03-04 EP claimed
WO-1991004016-A1 IMPLANTABLE DELIVERY DISPENSER ALZA CORPORATION (US) 1991-04-04 WO claimed
CN-1048327-A Contraceptive composition for male COHEN MICHAEL (NL) 1991-01-09 CN claimed
US-4252787-A CONTRACEPTIVES, PROGESTATIONAL ACTIVITY, STEROIDS CAMBRIDGE RESEARCH AND DEVELOPMENT GROUP (US) 1981-02-24 US claimed
US-4177269-A ANTITUMOR AGENTS AKTIEBOLAGET LEO (SE) 1979-12-04 US claimed
US-4018919-A IN MAMMALS ELI LILLY AND COMPANY (US) 1977-04-19 US claimed
US-4014987-A VAGINAL DEVICE; USING A HYDROPHOBIC POLYCARBOXYLIC ACID AS DRUG RELEASE RATE CONTROLLER ALZA CORPORATION (US) 1977-03-29 US claimed