SCHEMBL3751183

SCHEMBL3751183

COC(=O)OC(=O)c1cccnc1

nearest known ligand 0.74

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.74
KMT2A Q03164 8/20 0.58
MEN1 O00255 1/20 0.54
L3MBTL1 Q9Y468 1/20 0.53
APP P05067 1/20 0.52
GAA P10253 1/20 0.52
HCAR3 P49019 1/20 0.52
HCAR2 Q8TDS4 1/20 0.52
HDAC1 Q13547 1/20 0.51
HDAC6 Q9UBN7 1/20 0.51
MAPT P10636 1/20 0.51
HSD17B10 Q99714 1/20 0.51
LMNA P02545 3/20 0.50
THRB P10828 1/20 0.50
ATM Q13315 1/20 0.50
F7 P08709 1/20 0.50
F3 P13726 1/20 0.50
SARM1 Q6SZW1 1/20 0.50
SIRT2 Q8IXJ6 1/20 0.50
SIRT6 Q8N6T7 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10603067 0.89 ALDH1A1 (0.67) ALDH1A1KMT2AL3MBTL1APPGAA
SCHEMBL28309820 0.87 ALDH1A1 (0.65) ALDH1A1KMT2AL3MBTL1APPGAA
Methyl Nicotinate SCHEMBL820747 0.85 ALDH1A1 (1.00) ALDH1A1KMT2AL3MBTL1APPGAA
Methyl Nicotinate SCHEMBL24566 0.85 ALDH1A1 (1.00) ALDH1A1KMT2AL3MBTL1APPGAA
Methyl Nicotinate SCHEMBL29386553 0.85 ALDH1A1 (1.00) ALDH1A1KMT2AL3MBTL1APPGAA
SCHEMBL28520745 0.85 ALDH1A1 (0.62) ALDH1A1KMT2AL3MBTL1APPGAA
SCHEMBL31648307 0.85 ALDH1A1 (0.71) ALDH1A1KMT2AL3MBTL1APPGAA
SCHEMBL30659698 0.85 ALDH1A1 (0.71) ALDH1A1KMT2AL3MBTL1APPGAA
SCHEMBL2491556 0.85 ALDH1A1 (0.71) ALDH1A1KMT2AL3MBTL1APPGAA
Methyl Nicotinate SCHEMBL11491005 0.84 ALDH1A1 (0.96) ALDH1A1KMT2AL3MBTL1APPGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170058-A1 CETP INHIBITORS DERIVED FROM BENZOXAZOLE ARYLAMIDES Merck Sharp & Dohme Corp. (US) 2010-04-07 EP disclosed
WO-2008156715-A1 CETP INHIBITORS DERIVED FROM BENZOXAZOLE ARYLAMIDES MERCK & CO., INC. (US) 2008-12-24 WO disclosed
EP-1954287-A2 CETP INHIBITORS Merck & Co., Inc. (US) 2008-08-13 EP disclosed
WO-2007070173-A2 CETP INHIBITORS MERCK & CO., INC. (US) 2007-06-21 WO disclosed