SCHEMBL3755963

SCHEMBL3755963

O=C1[N]c2cc(NCCc3ccc(C(F)(F)F)cc3)ccc2N1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 3/20 0.42
CNR1 P21554 1/20 0.39
FFAR1 O14842 1/20 0.39
RORC P51449 1/20 0.39
MAPT P10636 2/20 0.39
KIF11 P52732 1/20 0.38
DAO P14920 1/20 0.38
PLAAT3 P53816 1/20 0.38
PLAAT5 Q96KN8 1/20 0.38
PLAAT2 Q9NWW9 1/20 0.38
PLAAT4 Q9UL19 1/20 0.38
CCNC P24863 1/20 0.37
CDK8 P49336 1/20 0.37
RXFP1 Q9HBX9 1/20 0.37
MCHR1 Q99705 1/20 0.37
PARP1 P09874 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TRPA1 O75762 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4752992 0.78 KIF11 (0.41) KIF11PARP1
SCHEMBL27791270 0.75 CNR1 (0.42) AURKBCNR1FFAR1RORCKIF11
SCHEMBL2234798 0.74 NTRK1 (0.47)
SCHEMBL1581297 0.73 FFAR1 (0.57) CNR1FFAR1RORCMAPTKIF11
SCHEMBL3804016 0.72 KMT2A (0.50) CNR1FFAR1MAPT
SCHEMBL3649276 0.71 RXFP1 (0.54) AURKBFFAR1MAPTCCNCCDK8
SCHEMBL6204891 0.71 MAPT (0.38) MAPTKIF11RXFP1SMN1; SMN2
SCHEMBL3644226 0.70 TAAR1 (0.49) CNR1FFAR1RORCMAPTPLAAT3
SCHEMBL3644611 0.69 ALDH1A1 (0.47) CNR1FFAR1RORCMAPTCCNC
SCHEMBL4750486 0.68 GRM2 (0.42) KIF11PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2185503-A1 MONOAMIDE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. Hoffmann-Roche AG (CH) 2010-05-19 EP disclosed
WO-2009016087-A1 MONOAMIDE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 2009-02-05 WO disclosed