SCHEMBL37583

SCHEMBL37583

Cc1cccc(Cc2nc3cc(C(=O)O)sc3c(=O)[nH]2)c1

nearest known ligand 0.78

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.78
CCNE1 P24864 4/20 0.44
CDK2 P24941 4/20 0.44
CDC7 O00311 3/20 0.44
ROCK1 Q13464 3/20 0.44
DBF4 Q9UBU7 3/20 0.44
KDM5B Q9UGL1 1/20 0.43
KMT2A Q03164 2/20 0.43
RNASEH1 O60930 2/20 0.43
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
CCNE2 O96020 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL37513 0.89 PDE5A (0.79) PDE5ACCNE1CDK2CDC7ROCK1
SCHEMBL38178 0.88 PDE5A (0.77) PDE5ACCNE1CDK2CDC7ROCK1
SCHEMBL37798 0.88 PDE5A (1.00) PDE5ACCNE1CDK2CDC7ROCK1
SCHEMBL38065 0.88 PDE5A (0.77) PDE5ACCNE1CDK2CDC7ROCK1
SCHEMBL37797 0.85 PDE5A (0.72) PDE5ACCNE1CDK2CDC7ROCK1
SCHEMBL38005 0.82 PDE5A (0.69) PDE5ACCNE1CDK2CDC7ROCK1
SCHEMBL3491573 0.82 PDE5A (0.78) PDE5ACCNE1CDK2KMT2ARNASEH1
SCHEMBL37942 0.81 PDE5A (0.78) PDE5AKMT2ARNASEH1KDM4E
SCHEMBL44227 0.81 PDE5A (0.67) PDE5ACCNE1CDK2CDC7ROCK1
SCHEMBL37981 0.81 PDE5A (0.66) PDE5ACCNE1CDK2CDC7ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004900-A1 THIENOPYRIMIDINE COMPOUNDS ASKA PHARMACEUTICAL CO., LTD. (JP) 2012-01-12 WO disclosed