SCHEMBL37797

SCHEMBL37797

O=C(O)c1cc2nc(Cc3cccc(C(F)(F)F)c3)[nH]c(=O)c2s1

nearest known ligand 0.72

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 3/20 0.72
CDC7 O00311 1/20 0.45
CCNE1 P24864 1/20 0.45
CDK2 P24941 1/20 0.45
ROCK1 Q13464 1/20 0.45
DBF4 Q9UBU7 1/20 0.45
GPR52 Q9Y2T5 4/20 0.42
KMT2A Q03164 2/20 0.42
DAO P14920 1/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL46031 0.87 PDE5A (0.56) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL38065 0.86 PDE5A (0.77) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL37513 0.85 PDE5A (0.79) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL37583 0.85 PDE5A (0.78) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL37798 0.84 PDE5A (1.00) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL38178 0.84 PDE5A (0.77) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL3493412 0.83 PDE5A (0.72) PDE5AGPR52KMT2ADAOALDH1A1
SCHEMBL44227 0.80 PDE5A (0.67) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL38005 0.79 PDE5A (0.69) PDE5ACDC7CCNE1CDK2ROCK1
SCHEMBL37942 0.78 PDE5A (0.78) PDE5AKMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012004900-A1 THIENOPYRIMIDINE COMPOUNDS ASKA PHARMACEUTICAL CO., LTD. (JP) 2012-01-12 WO disclosed
WO-2012004900-A1 THIENOPYRIMIDINE COMPOUNDS ASKA PHARMACEUTICAL CO., LTD. (JP) 2012-01-12 WO disclosed