SCHEMBL3767683

SCHEMBL3767683

C#Cc1cccc(C=O)c1-c1ncc[nH]1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.37
MTOR P42345 1/20 0.37
ADK P55263 1/20 0.37
ALDH1A1 P00352 3/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 1/20 0.33
CSNK1A1 P48729 1/20 0.33
TYRO3 Q06418 1/20 0.33
DYRK1B Q9Y463 1/20 0.33
TRIM24 O15164 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
KDM4E B2RXH2 2/20 0.32
IDO1 P14902 1/20 0.30
VCP P55072 1/20 0.30
ADRA2A P08913 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3767684 0.77 CSNK1A1 (0.41) NISCHMTORADKALDH1A1KMT2A
SCHEMBL3765764 0.71
SCHEMBL1663671 0.70 CSNK1A1 (0.53) NISCHMTORADKALDH1A1KMT2A
SCHEMBL38662055 0.70 CSNK1A1 (0.53) NISCHMTORADKALDH1A1KMT2A
SCHEMBL8596176 0.69 TAAR1 (0.39) NISCHMTORADKALDH1A1KMT2A
SCHEMBL711033 0.66 LMNA (0.55) ALDH1A1KMT2AMEN1TRIM24TRIM33
SCHEMBL9689968 0.66 KMT2A (0.42) ALDH1A1KMT2AMEN1TRIM24TRIM33
SCHEMBL6002606 0.66 ADRA2A (0.52) NISCHMTORADKALDH1A1KMT2A
Benzene SCHEMBL28197607 0.65 LMNA (0.52) ALDH1A1KMT2AMEN1TRIM24TRIM33
SCHEMBL11098154 0.65 NISCH (0.46) NISCHMTORADKALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193132-A2 3-SPIROPYRIMIDINETRIONE-QUINOLINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS AstraZeneca AB (SE) 2010-06-09 EP disclosed
WO-2009004382-A2 3-SPIROPYRIMIDINETRIONE-QUINOLINE DERIVATIVES AND THEIR USE AS ANTIBACTERIAL AGENTS ASTRAZENECA AB (SE) 2009-01-08 WO disclosed