Englitazone

Englitazone

SCHEMBL37697

O=C1NC(=O)C(Cc2ccc3c(c2)CCC(Cc2ccccc2)O3)S1

nearest known ligand 0.50

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PPARG P37231 4/20 0.50
FFAR1 O14842 7/20 0.47
ALDH1A1 P00352 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MAPT P10636 2/20 0.46
MAOB P27338 2/20 0.43
CA2 P00918 1/20 0.43
PPARA Q07869 2/20 0.43
PTPN1 P18031 1/20 0.42
MAOA P21397 2/20 0.42
CISD1 Q9NZ45 2/20 0.42
KDM4E B2RXH2 1/20 0.41
LMNA P02545 1/20 0.41
HIF1A Q16665 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Englitazone SCHEMBL20125577 1.00 PPARG (0.50) PPARGFFAR1ALDH1A1NPSR1MAPT
Englitazone SCHEMBL4727851 1.00 PPARG (0.50) PPARGFFAR1ALDH1A1NPSR1MAPT
Englitazone SCHEMBL20125579 1.00 PPARG (0.50) PPARGFFAR1ALDH1A1NPSR1MAPT
Englitazone SCHEMBL29377687 1.00 PPARG (0.50) PPARGFFAR1ALDH1A1NPSR1MAPT
Englitazone SCHEMBL9367929 0.99 PPARG (0.49) PPARGFFAR1ALDH1A1NPSR1MAPT
Englitazone SCHEMBL22607925 0.99 PPARG (0.49) PPARGFFAR1ALDH1A1NPSR1MAPT
Englitazone SCHEMBL8522765 0.99 PPARG (0.49) PPARGFFAR1ALDH1A1NPSR1MAPT
SCHEMBL9665642 0.92 FFAR1 (0.59) PPARGFFAR1ALDH1A1MAPTPPARA
SCHEMBL9664758 0.91 FFAR1 (0.58) PPARGFFAR1ALDH1A1MAPTPPARA
SCHEMBL6903859 0.89 PPARG (0.52) PPARGFFAR1ALDH1A1NPSR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 11466 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250360215-A1 PHARMACEUTICAL COMBINATIONS AND METHODS FOR PREVENTING OR TREATING NEURODEGENERATIVE DISEASES YUH CHIOU HWA (US) 2025-11-27 US claimed
US-20250332101-A1 Composition CORDEIRO MARIA FRANCESCA (GB) 2025-10-30 US claimed
EP-4640701-A2 GLUCAGON LIKE PEPTIDE 1 (GLP-1) FUSION PEPTIDE COUPLED CYCLIC PEPTIDE TYROSINE TYROSINE CONJUGATES AND USES THEREOF Janssen Sciences Ireland Unlimited Company (IE) 2025-10-29 EP claimed
US-20250281507-A1 METHODS OF TREATING NEPHROTIC SYNDROME THE RESEARCH INSTITUTE AT NATIONWIDE CHILDREN’S HOSPITAL 2025-09-11 US claimed
US-20250221962-A1 FABP4 AS A THERAPEUTIC TARGET IN SKIN DISEASES TICURE LTD (IL) 2025-07-10 US claimed
WO-2025136060-A1 CULTURE MEDIUM COMPOSITION FOR TRANSDIFFERENTIATION OF MUSCLE STEM CELLS INTO ADIPOCYTES, AND METHOD FOR PRODUCING CULTURED MEAT BY USING SAME 한화솔루션 주식회사 2025-06-26 WO claimed
CN-119698279-A Treatment of gastrointestinal disorders 阿克里普斯二有限公司 2025-03-25 CN claimed
CN-119613391-A Engliptin clean purification process 浙江大学衢州研究院 2025-03-14 CN claimed
EP-4520343-A2 GLUCAGON LIKE PEPTIDE 1 (GLP1)-GROWTH DIFFERENTIATION FACTOR 15 (GDF15) FUSION PROTEINS AND USES THEREOF Janssen Sciences Ireland Unlimited Company (IE) 2025-03-12 EP claimed
WO-2025049710-A1 PHARMACEUTICAL COMPOSITION FOR USE IN THE DISEASE TREATMENTS ACLIPSE TWO INC. (US) 2025-03-06 WO claimed
EP-0753298-A1 Synergistic combination comprising an insulin sensitizer and a HMG-CoA reductase inhibitor for treating arteriosclerosis SANKYO COMPANY LIMITED (JP) 1997-01-15 EP claimed
US-5594015-A Thiazolidine derivatives for the treatment of psoriasis REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1997-01-14 US claimed
CN-1134669-A Use of thiazolidinediones to prevent or delay onset of non-insulin dependent diabetes mellitus (NIDDM) SANKYO CO (JP) 1996-10-30 CN claimed
EP-0719140-A1 USE OF THIAZOLIDINEDIONES TO PREVENT OR DELAY ONSET OF NIDDM Sankyo Company Limited (JP) 1996-07-03 EP claimed
WO-1995035108-A1 THIAZOLIDINE DERIVATIVES FOR THE TREATMENT OF PSORIASIS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 1995-12-28 WO claimed
WO-1995007694-A1 USE OF THIAZOLIDINEDIONES TO PREVENT OR DELAY ONSET OF NIDDM SANKYO COMPANY, LIMITED (JP) 1995-03-23 WO claimed
EP-0207605-B1 HYPOGLYCEMIC THIAZOLIDINEDIONES PFIZER INC. (US) 1990-02-07 EP claimed
US-4703052-A Hypoglycemic thiazolidinediones PFIZER INC. (US) 1987-10-27 US claimed
EP-0207605-A1 Hypoglycemic thiazolidinediones PFIZER INC. (US) 1987-01-07 EP claimed
WO-1986007056-A1 HYPOGLYCEMIC THIAZOLIDINEDIONES PFIZER INC. (US) 1986-12-04 WO claimed