SCHEMBL3770108

SCHEMBL3770108

O=C1CCCN1c1ccccc1F

nearest known ligand 0.63

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.63
KMT2A Q03164 2/20 0.63
ALOX5AP P20292 1/20 0.47
FEN1 P39748 1/20 0.47
PARP1 P09874 2/20 0.45
MGLL Q99685 1/20 0.44
HSD17B10 Q99714 1/20 0.44
TP53 P04637 2/20 0.43
ALDH1A1 P00352 1/20 0.42
GFER P55789 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30157756 1.00 MEN1 (0.63) MEN1KMT2AALOX5APFEN1PARP1
SCHEMBL15108903 0.95 MEN1 (0.61) MEN1KMT2AALOX5APFEN1PARP1
SCHEMBL12478981 0.81 GFER (0.45) MEN1KMT2AALOX5APFEN1MGLL
SCHEMBL7787664 0.79 HSD17B10 (0.53) MEN1KMT2AALOX5APFEN1MGLL
SCHEMBL9360420 0.79 ADRA1B (0.51) PARP1HSD17B10TP53ALDH1A1
SCHEMBL22997585 0.78 HSD17B10 (0.44) MEN1KMT2AALOX5APFEN1MGLL
SCHEMBL5436101 0.78 ALOX5 (0.54) MGLLHSD17B10TP53ALDH1A1
SCHEMBL1901693 0.78 DDB1 (0.56) MEN1KMT2AHSD17B10
SCHEMBL3842955 0.78 HSD17B10 (0.44) MEN1KMT2AALOX5APFEN1MGLL
SCHEMBL8902463 0.78 NPC1 (0.49) MEN1KMT2AALOX5APFEN1MGLL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112262140-B Pesticidally active heterocyclic derivatives with sulfoximine containing substituents 先正达农作物保护股份公司 2024-05-28 CN disclosed
CN-109843886-A Two ring pyridone lactams and its application method 豪夫迈·罗氏有限公司 2019-06-04 CN disclosed
CN-103877080-B 4,5-bis-replaces-medicinal usage of 2-Pyrrolidone compound Key Laboratory of natural product chemistry, Chinese Academy of Sciences, Guizhou Province (CN) 2016-01-27 CN disclosed
CN-103877080-A New use of 4, 5-disubstituted-2-pyrrolidone compound KEY LAB OF CHEMISTRY NATURAL PRODUCTS OF GUIZHOU PROVINCE AND CHINESE ACADEMY 2014-06-25 CN disclosed
CN-101979378-B Method for synthesizing chiral gamma-lactam compounds SHANGHAI INST ORGANIC CHEM 2012-06-27 CN disclosed
CN-101979378-A Method for synthesizing chiral gamma-lactam compounds SHANGHAI INST ORGANIC CHEM 2011-02-23 CN disclosed
US-7846933-B2 such as 1-(4-Fluorophenyl)-5-(pyridin-4-yl)-4-imidazolin-2-one, having excellent p38 MAP kinase inhibitory action, useful for the treatment of osteoarthritis, arthritis, ulcerative colitis, Crohn's disease, psoriasis, dermatitis, asthma, bronchitis, pneumonia, rhinitis, conjunctivitis or keratitis MITSUBISHI TANABE PHARMA CORPORATION (JP) 2010-12-07 US disclosed
US-20090088422-A1 4-IMIDAZOLIN-2-ONE COMPOUNDS KUBO AKIRA 2009-04-02 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090088422-A1 4-IMIDAZOLIN-2-ONE COMPOUNDS OR10J3, NR4A3, NR3C2 MEN1 1829/4885KMT2A 1710/4885ALOX5AP 3790/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.