SCHEMBL3770851

SCHEMBL3770851

CC1CN(S(=O)(=O)c2ccc(C(F)(F)F)cc2)CCN1C(=O)c1cnn2cccnc12

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SPR P35270 1/20 0.43
HSD11B1 P28845 6/20 0.41
IDH1 O75874 1/20 0.41
KDM4E B2RXH2 1/20 0.40
SYK P43405 1/20 0.40
GAA P10253 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CNR1 P21554 1/20 0.39
IRAK4 Q9NWZ3 2/20 0.39
HDAC3 O15379 1/20 0.38
HDAC4 P56524 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC7 Q8WUI4 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC10 Q969S8 1/20 0.38
HDAC11 Q96DB2 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
HDAC9 Q9UKV0 1/20 0.38
HDAC5 Q9UQL6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL309552 1.00 SPR (0.43) SPRHSD11B1IDH1KDM4ESYK
SCHEMBL309343 1.00 SPR (0.43) SPRHSD11B1IDH1KDM4ESYK
SCHEMBL308921 0.89 PDE2A (0.48) SPRIDH1KDM4EGAANPSR1
SCHEMBL308584 0.89 PDE2A (0.48) SPRIDH1KDM4EGAANPSR1
SCHEMBL310252 0.88 SYK (0.43) SPRIDH1KDM4ESYKGAA
SCHEMBL308946 0.88 SYK (0.42) SPRIDH1KDM4ESYKGAA
SCHEMBL309128 0.86 PDE2A (0.40) SPRKDM4EGAAHDAC3HDAC4
SCHEMBL6411414 0.86 PDE2A (0.46) SPRALDH1A1
SCHEMBL6416356 0.85 HDAC3 (0.39) SPRKDM4EGAAHDAC3HDAC4
SCHEMBL309774 0.85 HDAC3 (0.41) SPRKDM4EGAAHDAC3HDAC4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2017046581-A1 COMPOSITION COMPRISING CAV2.2 CALCIUM CHANNEL BLOCKER AND OPIOID CALCHAN LIMITED (GB) 2017-03-23 WO disclosed
EP-2313413-B1 PYRAZOLO [1, 5-A] PYRIMIDINE DERIVATIVES CONVERGENCE PHARMACEUTICALS (GB) 2012-05-16 EP disclosed