SCHEMBL3780424

SCHEMBL3780424

CC(C)(C)OC(=O)N[C@@H](Cc1c[nH]nn1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ACE P12821 2/20 0.48
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
PTPN1 P18031 2/20 0.44
SCN9A Q15858 1/20 0.44
PPARA Q07869 8/20 0.44
PPARG P37231 7/20 0.44
IDO1 P14902 1/20 0.43
ITGA4 P13612 1/20 0.42
ITGB7 P26010 1/20 0.42
CTSS P25774 4/20 0.42
CTSK P43235 3/20 0.42
PPARD Q03181 2/20 0.42
CTSL P07711 1/20 0.42
CTSB P07858 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL304609 0.86 ITGA4 (0.39) ACEITGB3ITGA2BITGA4ITGB7
SCHEMBL304610 0.86 ITGA4 (0.39) ACEITGB3ITGA2BITGA4ITGB7
SCHEMBL28622648 0.85 PPARA (0.57) ACEITGB3ITGA2BPPARAPPARG
SCHEMBL28622647 0.85 PPARA (0.57) ACEITGB3ITGA2BPPARAPPARG
SCHEMBL13259431 0.83 TACR1 (0.52) ACEPPARACTSSCTSKCTSL
SCHEMBL1133305 0.82 ITGB3 (0.48) ACEITGB3ITGA2BPTPN1SCN9A
SCHEMBL214303 0.82 ITGB3 (0.48) ACEITGB3ITGA2BPTPN1SCN9A
SCHEMBL214302 0.82 ITGB3 (0.48) ACEITGB3ITGA2BPTPN1SCN9A
SCHEMBL18681589 0.81 CYP2D6 (0.40) CTSSCTSK
SCHEMBL29110986 0.79 ACE (0.51) ACEITGB3ITGA2BPTPN1SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2210882-A1 Synthesis of new protected azahistidine, their processes and their use in synthesises Commissariat à l'Énergie Atomique et aux Énergies Alternatives (FR) 2010-07-28 EP disclosed
WO-2010081882-A2 SYNTHESIS OF NEW PROTECTED AZAHISTIDINES, THEIR PROCESSES AND THEIR USE IN SYNTHESISES COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2010-07-22 WO disclosed