SCHEMBL3783903

SCHEMBL3783903

CCCC[Si](C)(C)OCCNc1ccnc2cc3c(cc12)OCO3

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 7/20 0.40
ADRA1D P25100 7/20 0.40
ADRA1A P35348 7/20 0.40
ADRA1B P35368 7/20 0.40
KDM4E B2RXH2 1/20 0.37
LMNA P02545 1/20 0.37
HTT P42858 1/20 0.37
HSD17B10 Q99714 1/20 0.37
CLK1 P49759 1/20 0.37
CCR1 P32246 1/20 0.37
EHMT2 Q96KQ7 2/20 0.37
EHMT1 Q9H9B1 2/20 0.37
FERMT2 Q96AC1 1/20 0.36
CDK1 P06493 1/20 0.36
CYP1A2 P05177 1/20 0.36
HPGD P15428 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4986900 0.85 HTR1A (0.49) HTR1AADRA1DADRA1AADRA1BCCR1
SCHEMBL527640 0.84 HTR1A (0.39) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL238033 0.81 HTR1A (0.41) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL3712435 0.81 CHRM2 (0.39) ADRA1DKDM4ELMNAHSD17B10HPGD
SCHEMBL13993581 0.78 PDE5A (0.44) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL241000 0.78 KDM4E (0.61) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL241926 0.77 HTR1A (0.40) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL241335 0.75 HTR1A (0.44) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL243582 0.75 FERMT2 (0.61) HTR1AADRA1DADRA1AADRA1BKDM4E
SCHEMBL241983 0.75 FERMT2 (0.51) HTR1AADRA1DADRA1AADRA1BKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010088544-A1 METHODS TO TREAT CANCER RUTGERS, THE STATE UNIVERSITY OF NEW JERSEY (US) 2010-08-05 WO disclosed