SCHEMBL3784136

SCHEMBL3784136

O=C1CCN(c2nc(NCc3ccccc3)nc3nnc(-c4ccc(F)cc4)nc23)CC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.44
PDE4B Q07343 2/20 0.44
PDE4C Q08493 2/20 0.44
PDE4D Q08499 2/20 0.44
HRH1 P35367 3/20 0.40
HRH4 Q9H3N8 3/20 0.40
MAPK13 O15264 1/20 0.39
MAPK12 P53778 1/20 0.39
MAPK11 Q15759 1/20 0.39
MAPK14 Q16539 1/20 0.39
TP53 P04637 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KCNH3 Q9ULD8 2/20 0.38
GPR68 Q15743 2/20 0.38
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
HRH2 P25021 1/20 0.37
HRH3 Q9Y5N1 1/20 0.37
TLR9 Q9NR96 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3785003 0.87 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3779641 0.87 HTT (0.50) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL3704626 0.87 HRH4 (0.52) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3786948 0.86 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3784610 0.85 PDE4A (0.50) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3788927 0.85 ACHE (0.44) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3783454 0.84 ACHE (0.47) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3781421 0.83 PDE4A (0.41) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3702614 0.82 HTT (0.42) PDE4APDE4BPDE4CPDE4DHRH1
SCHEMBL3781010 0.82 HRH4 (0.52) PDE4APDE4BPDE4CPDE4DHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed