SCHEMBL3781421

SCHEMBL3781421

Fc1ccc(-c2nnc3nc(NCc4ccccc4)nc(N4CCC(NC5CCCCC5)CC4)c3n2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 2/20 0.41
PDE4B Q07343 2/20 0.41
PDE4C Q08493 2/20 0.41
PDE4D Q08499 2/20 0.41
TLR9 Q9NR96 2/20 0.39
TLR7 Q9NYK1 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
OPRK1 P41145 7/20 0.38
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP2D6 P10635 1/20 0.37
HTT P42858 1/20 0.37
HRH4 Q9H3N8 2/20 0.36
HRH1 P35367 1/20 0.36
CTNNB1 P35222 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3783454 0.89 ACHE (0.47) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3786948 0.87 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3781745 0.85 ACHE (0.38) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3704323 0.85 CCNE2 (0.40) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3701586 0.83 TLR9 (0.39) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3779641 0.83 HTT (0.50) PDE4APDE4BPDE4CPDE4DACHE
SCHEMBL3704626 0.83 HRH4 (0.52) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3785003 0.83 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3784136 0.83 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DTLR9
SCHEMBL3788927 0.81 ACHE (0.44) PDE4APDE4BPDE4CPDE4DTLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO claimed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed