SCHEMBL3779641

SCHEMBL3779641

Fc1ccc(-c2nnc3nc(NCc4ccccc4)nc(N4CCOCC4)c3n2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
PDE4A P27815 3/20 0.46
PDE4B Q07343 3/20 0.46
PDE4C Q08493 3/20 0.46
PDE4D Q08499 3/20 0.46
LMNA P02545 4/20 0.46
GAA P10253 2/20 0.46
ALDH1A1 P00352 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PIK3CB P42338 4/20 0.45
TSHR P16473 2/20 0.45
PKM P14618 2/20 0.45
CRHBP P24387 1/20 0.45
CRHR2 Q13324 1/20 0.45
GLA P06280 1/20 0.44
KDM4E B2RXH2 2/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
HPGD P15428 1/20 0.43
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3702614 0.95 HTT (0.42) HTTPDE4APDE4BPDE4CPDE4D
SCHEMBL3785003 0.88 PDE4A (0.47) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL3704626 0.88 HRH4 (0.52) PDE4APDE4BPDE4CPDE4DALDH1A1
SCHEMBL3784136 0.87 PDE4A (0.44) PDE4APDE4BPDE4CPDE4DSMN1; SMN2
SCHEMBL3786948 0.87 PDE4A (0.43) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL3779078 0.86 MTOR (0.42) PIK3CA
SCHEMBL13286093 0.86 TLR9 (0.44) PDE4APDE4BPDE4CPDE4DPIK3CA
SCHEMBL3788927 0.86 ACHE (0.44) PDE4APDE4BPDE4CPDE4DLMNA
SCHEMBL3783454 0.85 ACHE (0.47) PDE4APDE4BPDE4CPDE4DMEN1
SCHEMBL3777960 0.85 GHSR (0.40) LMNAALDH1A1MEN1KMT2APIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO claimed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed