SCHEMBL3784417

SCHEMBL3784417

COc1ccc(Cn2cc(C[C@H](NC(=O)OC(C)(C)C)C(=O)O)nn2)cc1

nearest known ligand 0.52

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PPARA Q07869 3/20 0.52
PPARG P37231 2/20 0.52
KDM1A O60341 1/20 0.51
HDAC1 Q13547 1/20 0.49
ITGB3 P05106 1/20 0.48
ITGA2B P08514 1/20 0.48
ITGA4 P13612 2/20 0.47
ITGB7 P26010 2/20 0.47
PTPN1 P18031 5/20 0.47
ACE P12821 1/20 0.46
CYP19A1 P11511 2/20 0.46
CDC25B P30305 3/20 0.46
PTPN2 P17706 2/20 0.46
CDC25A P30304 1/20 0.46
MEN1 O00255 1/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3331695 0.91 ACE (0.56) PPARAPPARGPTPN1ACECDC25B
SCHEMBL304588 0.91 ACE (0.56) PPARAPPARGPTPN1ACECDC25B
SCHEMBL3789613 0.90 HDAC1 (0.49) PPARAPPARGKDM1AHDAC1ITGB3
SCHEMBL26347313 0.84 ACE (0.49) PPARAPPARGKDM1AITGB3ITGA2B
SCHEMBL29034539 0.84 ACE (0.49) PPARAPPARGKDM1AITGB3ITGA2B
SCHEMBL305197 0.82 CYP19A1 (0.49) HDAC1CYP19A1
SCHEMBL335310 0.81 ITGB3 (0.67) PPARAPPARGITGB3ITGA2BITGA4
SCHEMBL335309 0.81 ITGB3 (0.67) PPARAPPARGITGB3ITGA2BITGA4
SCHEMBL1308867 0.81 ITGB3 (0.67) PPARAPPARGITGB3ITGA2BITGA4
SCHEMBL756405 0.81 PTPN1 (0.49) PPARAPPARGPTPN1ACECDC25B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2210882-A1 Synthesis of new protected azahistidine, their processes and their use in synthesises Commissariat à l'Énergie Atomique et aux Énergies Alternatives (FR) 2010-07-28 EP disclosed
WO-2010081882-A2 SYNTHESIS OF NEW PROTECTED AZAHISTIDINES, THEIR PROCESSES AND THEIR USE IN SYNTHESISES COMMISSARIAT A L'ENERGIE ATOMIQUE ET AUX ENERGIES ALTERNATIVES (FR) 2010-07-22 WO disclosed