SCHEMBL3784769

SCHEMBL3784769

CNS(=O)(=O)c1ccc(CNc2ncc3c(n2)NNC(c2ccc(F)cc2)=N3)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 10/20 0.44
PTGS1 P23219 1/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
GAA P10253 2/20 0.39
MEN1 O00255 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
ALOX12 P18054 1/20 0.39
CYP2C19 P33261 1/20 0.39
HTT P42858 1/20 0.39
GFER P55789 1/20 0.39
KMT2A Q03164 1/20 0.39
KIT P10721 1/20 0.38
VNN1 O95497 1/20 0.37
TP53 P04637 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
CCR1 P32246 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3781294 0.88 PTGS2 (0.46) PTGS2
SCHEMBL3783206 0.88 KDM4E (0.42) PTGS2KDM4EALDH1A1GAAMEN1
SCHEMBL3785754 0.82 PTGS2 (0.46) PTGS2KDM4EALDH1A1GAAMEN1
SCHEMBL3778909 0.79 ALDH1A1 (0.44) ALDH1A1MEN1CYP1A2CYP2D6CYP2C9
SCHEMBL3789005 0.78 MAPT (0.46) KDM4EALDH1A1GAAMEN1HPGD
SCHEMBL3783814 0.75 MERTK (0.45)
SCHEMBL3781754 0.73 PTGS2 (0.46) PTGS2PTGS1KDM4EALDH1A1GAA
SCHEMBL3706406 0.69 KDM4E (0.41) PTGS2KDM4EALDH1A1GAAMEN1
SCHEMBL3794400 0.69 USP2 (0.44) PTGS2CYP1A2CYP2C9CYP2C19TSHR
SCHEMBL3788169 0.67 MAPT (0.48) KDM4EALDH1A1CYP1A2CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO claimed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed