SCHEMBL3785754

SCHEMBL3785754

Fc1ccc(C2=Nc3cnc(NCc4ccccc4)nc3NN2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 1/20 0.46
TP53 P04637 3/20 0.46
GAA P10253 3/20 0.46
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
ALOX15 P16050 1/20 0.46
TSHR P16473 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
KCNH3 Q9ULD8 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
LMNA P02545 2/20 0.39
HPGD P15428 2/20 0.38
MAPK14 Q16539 4/20 0.38
MAPK13 O15264 3/20 0.38
MAPK12 P53778 3/20 0.38
MAPK11 Q15759 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3783206 0.94 KDM4E (0.42) PTGS2TP53GAAKDM4EALDH1A1
SCHEMBL3778909 0.84 ALDH1A1 (0.44) TP53ALDH1A1ALOX15TSHRMAPK1
SCHEMBL3781294 0.84 PTGS2 (0.46) PTGS2
SCHEMBL3794400 0.83 USP2 (0.44) PTGS2TSHRMAPK1KCNH3LMNA
SCHEMBL3784769 0.82 PTGS2 (0.44) PTGS2TP53GAAKDM4EALDH1A1
SCHEMBL3789005 0.81 MAPT (0.46) TP53GAAKDM4EALDH1A1MAPK1
SCHEMBL3788169 0.81 MAPT (0.48) TP53KDM4EALDH1A1L3MBTL1SMN1; SMN2
SCHEMBL3783814 0.81 MERTK (0.45) KCNH3
SCHEMBL3706406 0.74 KDM4E (0.41) PTGS2TP53GAAKDM4EALDH1A1
SCHEMBL3780214 0.73 ADORA1 (0.41) GAAKDM4EALDH1A1SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed
WO-2010083645-A1 PYRIMIDO[5,4-e][1,2,4]TRIAZINES AND USES THEREOF SHANGHAI TARGETDRUG CO., LTD (CN) 2010-07-29 WO disclosed