SCHEMBL3785356

SCHEMBL3785356

COC(=O)c1ccc2c(C3CCCCC3)c(Br)[nH]c2c1.COCOc1c(C)cccc1-c1[nH]c2cc(C(=O)OC)ccc2c1C1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 2/20 0.39
KIF11 P52732 1/20 0.38
ALDH1A1 P00352 3/20 0.36
MAPK1 P28482 1/20 0.36
DYRK1A Q13627 1/20 0.35
GSK3B P49841 2/20 0.34
HPGD P15428 2/20 0.34
PTPN1 P18031 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34
GAA P10253 2/20 0.33
HSD17B10 Q99714 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
PKM P14618 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2275400 0.95 PARP1 (0.42) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL3787651 0.85 ALDH1A1 (0.41) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL3787653 0.85 ALDH1A1 (0.41) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL4562814 0.82 PARP1 (0.45) PARP1KIF11ALDH1A1MAPK1GSK3B
SCHEMBL3793445 0.81 PARP1 (0.47) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL50237 0.81 PARP1 (0.50) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL1173615 0.80 KIF11 (0.51) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL5283403 0.79 PARP1 (0.44) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL772671 0.77 EGFR (0.41) PARP1KIF11ALDH1A1MAPK1DYRK1A
SCHEMBL2273262 0.77 EGFR (0.41) PARP1KIF11ALDH1A1MAPK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010082050-A1 MACROCYCLIC AND 7-AMINOALKYL-SUBSTITUTED BENZOXAZOCINES FOR TREATMENT OF HEPATITIS C INFECTIONS ISTITUTO DI RICERCHE DI BIOLOGIA MOLECOLARE P. ANGELETTI S.P.A. (IT) 2010-07-22 WO disclosed