SCHEMBL3785605

SCHEMBL3785605

O=C(Nc1ccc(F)cc1)c1ccc(N2CCc3ccccc3C2)nc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.58
KMT2A Q03164 2/20 0.58
MEN1 O00255 1/20 0.58
TNF P01375 1/20 0.58
NOD2 Q9HC29 1/20 0.58
NOD1 Q9Y239 1/20 0.58
CYP1A2 P05177 2/20 0.54
CYP3A4 P08684 2/20 0.54
CYP2D6 P10635 2/20 0.54
CYP2C19 P33261 2/20 0.54
CYP2C9 P11712 1/20 0.54
NPC1 O15118 1/20 0.53
GRIN2D O15399 4/20 0.50
GRIN3B O60391 4/20 0.50
GRIN1 Q05586 4/20 0.50
GRIN2A Q12879 4/20 0.50
GRIN2B Q13224 4/20 0.50
GRIN2C Q14957 4/20 0.50
GRIN3A Q8TCU5 4/20 0.50
NAMPT P43490 2/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3793530 0.91 PTPN11 (0.58) RAB9AKMT2AMEN1NPC1GRIN2D
SCHEMBL3796116 0.85 MAPT (0.59) RAB9AKMT2AMEN1TNFNOD2
SCHEMBL3788726 0.83 GRIN2D (0.54) RAB9AKMT2AMEN1NPC1GRIN2D
SCHEMBL13203909 0.83 GRIN2D (0.61) RAB9AKMT2AMEN1NPC1GRIN2D
SCHEMBL3794388 0.82 KDM4E (0.60) RAB9AKMT2ANPC1GRIN2DGRIN3B
SCHEMBL3783683 0.81 GRIN2D (0.55) RAB9AKMT2AMEN1NPC1GRIN2D
SCHEMBL3063610 0.81 ALDH1A1 (0.60) RAB9AKMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3058918 0.81 RAB9A (0.72) RAB9AKMT2ACYP1A2CYP3A4CYP2D6
SCHEMBL3788716 0.80 SMN1; SMN2 (0.58) KMT2AMEN1GRIN2DGRIN3BGRIN1
SCHEMBL3788319 0.80 KDM4E (0.59) RAB9AKMT2AMEN1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO claimed
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO disclosed
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO disclosed