SCHEMBL3794388

SCHEMBL3794388

COc1cccc(NC(=O)c2ccc(N3CCc4ccccc4C3)nc2)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.60
HPGD P15428 1/20 0.60
RAB9A P51151 5/20 0.58
NPC1 O15118 4/20 0.58
PDGFRB P09619 1/20 0.55
KDR P35968 1/20 0.55
TP53 P04637 2/20 0.52
SMN1; SMN2 Q16637 3/20 0.51
NLRP3 Q96P20 1/20 0.51
ALDH1A1 P00352 1/20 0.51
PKM P14618 1/20 0.51
KMT2A Q03164 1/20 0.51
TSHR P16473 1/20 0.51
GRIN2D O15399 1/20 0.51
GRIN3B O60391 1/20 0.51
GRIN1 Q05586 1/20 0.51
GRIN2A Q12879 1/20 0.51
GRIN2B Q13224 1/20 0.51
GRIN2C Q14957 1/20 0.51
GRIN3A Q8TCU5 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3793530 0.86 PTPN11 (0.58) KDM4ERAB9ANPC1KDRTP53
SCHEMBL3796116 0.85 MAPT (0.59) KDM4ERAB9ASMN1; SMN2ALDH1A1KMT2A
SCHEMBL2305301 0.85 GRIN2D (0.51) PDGFRBKDRSMN1; SMN2GRIN2DGRIN3B
SCHEMBL3794970 0.84 NAMPT (0.58) KDM4ERAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL3788319 0.83 KDM4E (0.59) KDM4EHPGDRAB9ANPC1TP53
SCHEMBL3785605 0.82 RAB9A (0.58) RAB9ANPC1SMN1; SMN2KMT2AGRIN2D
SCHEMBL6140213 0.80 KDM4E (0.62) KDM4EHPGDRAB9ANPC1TP53
SCHEMBL3796096 0.80 PRMT5 (0.52) RAB9ANPC1SMN1; SMN2KMT2AGRIN2D
SCHEMBL2302759 0.80 KDM4E (0.61) KDM4EHPGDRAB9ANPC1TP53
SCHEMBL3788726 0.78 GRIN2D (0.54) RAB9ANPC1SMN1; SMN2KMT2AGRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO claimed
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO disclosed
WO-2010143803-A2 NEW NICOTINAMIDE DERIVATIVES WITH ANTI-ANDROGEN EFFECTS, PROCESSES OF PREPARING, AND ANTIANDROGENS COMPRISING THE SAME INDUSTRY FOUNDATION OF CHONNAM NATIONAL UNIVERSITY (KR) 2010-12-16 WO disclosed