SCHEMBL3785957

SCHEMBL3785957

O=C(Oc1ccccn1)C1CCN(C(=O)O)CC1

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 1/20 0.44
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 2/20 0.42
CYP2C19 P33261 2/20 0.41
NPC1 O15118 3/20 0.41
RAB9A P51151 3/20 0.41
POLB P06746 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 2/20 0.40
TSHR P16473 1/20 0.39
RIPK1 Q13546 1/20 0.39
NOS2 P35228 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20558297 0.85 KMT2A (0.46) L3MBTL1NPC1RAB9APOLBSMN1; SMN2
SCHEMBL3804900 0.82 GPR119 (0.60) POLBKDM4E
SCHEMBL28737837 0.81 SMN1; SMN2 (0.51) ALDH1A1L3MBTL1RAB9APOLBSMN1; SMN2
SCHEMBL5152829 0.80 EPHX2 (0.63) EPHX2RIPK1
SCHEMBL2474885 0.80 KMT2A (0.42) L3MBTL1NPC1RAB9APOLBSMN1; SMN2
Hydrochloric Acid SCHEMBL23928369 0.79 EPHX2 (0.62) EPHX2RIPK1
SCHEMBL30473865 0.78 L3MBTL1 (0.40) L3MBTL1RAB9APOLBSMN1; SMN2
SCHEMBL28987117 0.77 CYP2C19 (0.46) ALDH1A1L3MBTL1CYP2C19NPC1POLB
Hydrochloric Acid SCHEMBL27414475 0.77 PKM (0.39) L3MBTL1RAB9APOLBSMN1; SMN2
SCHEMBL440330 0.75 CYP3A4 (0.54) EPHX2ALDH1A1L3MBTL1CYP2C19POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2398796-A1 HETEROCYCLIC DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE Merck Canada Inc. (CA) 2011-12-28 EP disclosed
WO-2010094126-A1 HETEROCYCLIC DERIVATIVES AS INHIBITORS OF STEAROYL-COENZYME A DELTA-9 DESATURASE MERCK FROSST CANADA LTD. (CA) 2010-08-26 WO disclosed