SCHEMBL3786153

SCHEMBL3786153

COc1ccc(-c2[nH]c(=O)cc(-c3ccccc3)c2-c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.56
KDM4E B2RXH2 3/20 0.56
SMN1; SMN2 Q16637 2/20 0.56
HPGD P15428 1/20 0.56
PTGS2 P35354 2/20 0.48
BACE1 P56817 3/20 0.48
HDAC4 P56524 1/20 0.48
HDAC2 Q92769 1/20 0.48
HDAC8 Q9BY41 1/20 0.48
MAPT P10636 2/20 0.46
PTGS1 P23219 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MAP2K1 Q02750 1/20 0.45
ABL1 P00519 1/20 0.45
ABCB1 P08183 1/20 0.45
BCR P11274 1/20 0.45
PDE10A Q9Y233 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3796574 0.83 PTGS2 (0.46) ALDH1A1KDM4ESMN1; SMN2HPGDPTGS2
SCHEMBL3789193 0.80 PTGS2 (0.45) ALDH1A1KDM4ESMN1; SMN2HPGDPTGS2
SCHEMBL1573422 0.78 KDM4E (0.50) ALDH1A1KDM4EHPGDPTGS2BACE1
SCHEMBL20323146 0.77 BACE1 (0.59) ALDH1A1KDM4ESMN1; SMN2HPGDPTGS2
SCHEMBL7093922 0.75 ALDH1A1 (0.51) ALDH1A1KDM4ESMN1; SMN2HPGDPTGS2
SCHEMBL5904146 0.74 PDE10A (0.60) ALDH1A1KDM4EMAPTKMT2AMAP2K1
SCHEMBL7039067 0.74 PTGS2 (0.72) ALDH1A1KDM4ESMN1; SMN2HPGDPTGS2
SCHEMBL28260523 0.74 GCGR (0.64) ALDH1A1KDM4ESMN1; SMN2MAPTMEN1
SCHEMBL7042910 0.74 PTGS2 (0.72) ALDH1A1KDM4ESMN1; SMN2HPGDPTGS2
SCHEMBL15057905 0.73 PTGS2 (0.60) ALDH1A1KDM4EHPGDPTGS2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010093595-A1 FUNGICIDAL 2-PYRIDONES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2010-08-19 WO claimed
WO-2010093595-A1 FUNGICIDAL 2-PYRIDONES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2010-08-19 WO disclosed