SCHEMBL378787

SCHEMBL378787

O=C(CCC(=O)Oc1ccc2ccc3ccccc3c2c1)Oc1ccc2ccc3ccccc3c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.51
CYP1A2 P05177 3/20 0.51
KMT2A Q03164 3/20 0.51
MEN1 O00255 2/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
TDP1 Q9NUW8 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 2/20 0.46
PDGFRB P09619 2/20 0.46
PDGFRA P16234 2/20 0.46
HSD17B10 Q99714 3/20 0.46
MAPT P10636 3/20 0.46
LMNA P02545 1/20 0.46
HTT P42858 1/20 0.46
HIF1A Q16665 2/20 0.45
CYP1B1 Q16678 1/20 0.45
SIRT5 Q9NXA8 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL378788 0.94 CYP1A2 (0.52) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL15882797 0.92 PDGFRB (0.55) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL28010902 0.90 TDP1 (0.47) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL15882772 0.88 PDGFRB (0.49) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL31482564 0.87 TDP1 (0.44) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL34462112 0.87 TDP1 (0.44) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL30859625 0.87 KMT2A (0.44) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL28010903 0.85 CYP1A2 (0.47) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL31634147 0.84 SIRT5 (0.47) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2
SCHEMBL25210358 0.83 PDGFRB (0.46) ALDH1A1CYP1A2KMT2AMEN1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408791-A1 FOSFLUCONAZOLE DERIVATIVES, SYNTHESIS, AND USE IN LONG ACTING FORMULATIONS SEPS Pharma N.V. (BE) 2012-01-25 EP disclosed
WO-2010105910-A1 FOSFLUCONAZOLE DERIVATIVES, SYNTHESIS, AND USE IN LONG ACTING FORMULATIONS SEPS PHARMA N.V. (BE) 2010-09-23 WO disclosed