SCHEMBL3788071

SCHEMBL3788071

COc1ccccc1CCNC(=O)c1ccc2c(c1)CCCO2

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.58
MAPT P10636 4/20 0.56
MEN1 O00255 1/20 0.56
KMT2A Q03164 1/20 0.56
NPC1 O15118 5/20 0.55
RAB9A P51151 3/20 0.55
NAMPT P43490 1/20 0.54
PAX8 Q06710 2/20 0.53
KLF5 Q13887 2/20 0.53
POLB P06746 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
PKM P14618 1/20 0.52
PTGDR2 Q9Y5Y4 1/20 0.51
ROCK2 O75116 1/20 0.51
ROCK1 Q13464 1/20 0.51
HPGD P15428 2/20 0.49
CTNNB1 P35222 2/20 0.49
WNT3A P56704 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.49
MTNR1A P48039 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3787714 0.81 HPGD (0.54) MAPTNPC1RAB9APAX8KLF5
SCHEMBL1569557 0.75 PTGDR2 (0.69) PTGDR2
SCHEMBL15979797 0.74 CTNNB1 (0.84) CTNNB1WNT3A
SCHEMBL29111414 0.74 MTNR1A (0.65) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL26115654 0.73 KDM4E (0.68) MAPTNPC1RAB9APAX8KLF5
SCHEMBL8882813 0.73 MEN1 (0.52) TAAR1MAPTMEN1KMT2ANPC1
SCHEMBL3787786 0.72 TAS1R3 (0.61) NPC1RAB9AROCK2ROCK1CTNNB1
SCHEMBL8317337 0.72 CTNNB1 (0.56) KMT2ANPC1RAB9APAX8KLF5
SCHEMBL28860886 0.72 CTNNB1 (0.60) KMT2ANPC1RAB9ACTNNB1WNT3A
SCHEMBL671055 0.72 CTNNB1 (0.57) NPC1RAB9ATDP1CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234486-A1 BENZIMIDAZOLES AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079011-A1 BENZIMIDAZOLES AND ANALOGS AS RHO KINASE INHIBITORS THE SCRIPPS RESEARCH INSTITUTE (US) 2009-06-25 WO disclosed