SCHEMBL3790116

SCHEMBL3790116

O=C(NCc1ccccc1OC(F)(F)F)c1ccc2nn(Cc3ccccn3)c(=O)n2c1

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 9/20 0.47
RIPK1 Q13546 3/20 0.45
HSD17B13 Q7Z5P4 3/20 0.45
ROCK2 O75116 2/20 0.44
ROCK1 Q13464 1/20 0.44
PPARG P37231 2/20 0.43
CYP2C9 P11712 1/20 0.42
CYP2J2 P51589 1/20 0.42
HDAC3 O15379 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13257878 0.90 EPHX2 (0.41) EPHX2RIPK1HSD17B13ROCK2ROCK1
SCHEMBL3792366 0.89 EPHX2 (0.49) EPHX2ROCK2ROCK1
SCHEMBL3787484 0.88 EPHX2 (0.39) EPHX2RIPK1HSD17B13ROCK2ROCK1
Hydrochloric Acid SCHEMBL3792564 0.88 EPHX2 (0.39) EPHX2RIPK1HSD17B13ROCK2ROCK1
SCHEMBL3787655 0.87 ROCK2 (0.48) EPHX2RIPK1HSD17B13ROCK2ROCK1
SCHEMBL3796727 0.86 EPHX2 (0.52) EPHX2RIPK1HSD17B13ROCK2ROCK1
SCHEMBL3791214 0.86 EPHX2 (0.45) EPHX2RIPK1HSD17B13ROCK2ROCK1
Sulfuric Acid SCHEMBL3794696 0.86 EPHX2 (0.38) EPHX2RIPK1HSD17B13ROCK2ROCK1
SCHEMBL13258052 0.86 EPHX2 (0.49) EPHX2RIPK1HSD17B13ROCK2ROCK1
SCHEMBL3790889 0.86 PPARG (0.52) EPHX2RIPK1HSD17B13ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed
WO-2010096722-A1 3-OXO-2, 3-DIHYDRO- [1,2, 4] TRIAZOLO [4, 3-A]PYRIDINES AS SOLUBLE EPOXIDE HYDROLASE (SEH) INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-08-26 WO disclosed