SCHEMBL379032

SCHEMBL379032

Cc1noc(-c2ccc(C(=O)N3CCC(C(=O)O)(c4ccc(F)cc4)CC3)cc2)n1.O=C(c1ccc(-c2ccc(F)cc2)cc1)N1CCC(C(=O)NC(CC2CC2)c2ccccc2)(c2ccc(F)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
IDO1 P14902 1/20 0.37
TACR3 P29371 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD11B1 P28845 1/20 0.36
TACR1 P25103 1/20 0.35
PTPN2 P17706 1/20 0.35
PTPN1 P18031 1/20 0.35
OPRL1 P41146 1/20 0.35
NPY2R P49146 1/20 0.35
CCR5 P51681 1/20 0.35
ABCC3 O15438 1/20 0.34
ABCC4 O15439 1/20 0.34
ABCB11 O95342 1/20 0.34
CYP2C8 P10632 1/20 0.34
ABCB4 P21439 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3721822 0.97 ADRB3 (0.40) ADRB3SLC6A2SLC6A4IDO1TACR3
SCHEMBL3721825 0.88 ADRB3 (0.39) ADRB3SLC6A2SLC6A4IDO1TACR3
SCHEMBL7908350 0.87 HSD11B1 (0.46) SLC6A4HSD11B1TACR1PTPN1OPRL1
SCHEMBL13092251 0.85 BDKRB1 (0.40) ADRB3SLC6A2SLC6A4IDO1TACR3
SCHEMBL396983 0.84 TACR1 (0.40) ADRB3SLC6A2SLC6A4TACR3CYP2C9
SCHEMBL379339 0.83 TSHR (0.42) ADRB3SLC6A2SLC6A4TACR3NPY2R
SCHEMBL378186 0.83 TACR3 (0.46) IDO1TACR3CYP2C9CYP1A2CYP2C19
SCHEMBL437707 0.83 HSD11B1 (0.41) SLC6A4HSD11B1TACR1PTPN1OPRL1
SCHEMBL378669 0.82 TACR1 (0.41) SLC6A4TACR3CYP2C9CYP1A2CYP2C19
SCHEMBL13092448 0.81 IDO1 (0.39) ADRB3SLC6A2SLC6A4IDO1TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP claimed