SCHEMBL396983

SCHEMBL396983

C[C@H](NC(=O)C1(c2ccccc2)CCN(C(=O)c2ccc(-c3ccc(F)cc3)cc2)CC1)c1ccccc1.Cc1noc(-c2ccc(C(=O)N3CCC(C(=O)N[C@@H](C)c4ccccc4)(c4ccccc4)CC3)cc2)n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 1/20 0.40
TSHR P16473 2/20 0.40
BDKRB1 P46663 2/20 0.40
TACR3 P29371 2/20 0.39
SCD5 Q86SK9 1/20 0.39
NPC1 O15118 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SLC6A4 P31645 2/20 0.39
NPY2R P49146 1/20 0.39
NPY1R P25929 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
SLC6A7 Q99884 1/20 0.38
ATM Q13315 1/20 0.38
ALDH1A1 P00352 1/20 0.38
LMNA P02545 1/20 0.38
HSD11B1 P28845 1/20 0.37
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13092251 0.98 BDKRB1 (0.40) TACR1TSHRBDKRB1TACR3SCD5
SCHEMBL378669 0.98 TACR1 (0.41) TACR1TSHRBDKRB1TACR3SCD5
SCHEMBL378915 0.95 TSHR (0.43) TSHRBDKRB1SCD5NPC1SLC6A4
SCHEMBL379355 0.94 TACR3 (0.41) TACR1BDKRB1TACR3CYP1A2CYP2C9
SCHEMBL378830 0.91 BDKRB1 (0.42) TACR1BDKRB1TACR3CYP1A2CYP2C9
SCHEMBL13092272 0.90 TACR3 (0.42) TSHRBDKRB1TACR3SCD5NPC1
SCHEMBL395363 0.89 THRB (0.43) TACR1TSHRBDKRB1SCD5CYP2C9
SCHEMBL13092261 0.88 ALDH1A1 (0.42) TSHRBDKRB1SCD5SLC6A4ATM
SCHEMBL3714839 0.88 NPC1 (0.49) TACR1TSHRNPC1CYP2C9CYP2C19
SCHEMBL7908720 0.88 CTSL (0.42) TACR1TSHRBDKRB1TACR3SCD5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2408745-A1 PIPERIDINE DERIVATIVES AS NK3 RECEPTOR ANTAGONISTS F. Hoffmann-La Roche AG (CH) 2012-01-25 EP disclosed