SCHEMBL3794485

SCHEMBL3794485

Cc1c(CNc2ccc3c(c2)O[C@H](C)[CH]3)cccc1-n1c(C2CCCO2)nc2cc(C(F)(F)F)ccc21

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DHFR P00374 1/20 0.33
GAA P10253 1/20 0.31
PIK3CA P42336 1/20 0.31
PIK3CB P42338 1/20 0.31
PIK3CG P48736 1/20 0.31
USP2 O75604 1/20 0.30
PKM P14618 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3791360 0.91 DHFR (0.34) DHFR
SCHEMBL3794538 0.90 CYP2D6 (0.32) DHFR
SCHEMBL3791152 0.89 DHFR (0.34) DHFRGAAPKM
SCHEMBL3795976 0.89 PDE10A (0.34) DHFRGAA
SCHEMBL3795926 0.86 NPC1 (0.37) GAAPIK3CAPIK3CBPIK3CGUSP2
SCHEMBL1708131 0.83 FFAR1 (0.38) USP2PKM
SCHEMBL10292325 0.83 FFAR1 (0.38) USP2PKM
SCHEMBL10291346 0.82 LMNA (0.39) USP2PKM
SCHEMBL1708368 0.82 LMNA (0.33) GAAPIK3CAPIK3CBPIK3CGUSP2
SCHEMBL1707938 0.81 DHFR (0.39) DHFRPIK3CAPIK3CBPIK3CGUSP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed