SCHEMBL3795994

SCHEMBL3795994

NC(=O)c1cnc(NCc2ccc3c(c2)OCO3)nc1

nearest known ligand 0.76

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC3 O15379 1/20 0.76
HDAC1 Q13547 1/20 0.76
HDAC2 Q92769 1/20 0.76
HDAC6 Q9UBN7 1/20 0.76
PDE5A O76074 2/20 0.61
AURKA O14965 2/20 0.55
RPS6KB1 P23443 2/20 0.55
AURKB Q96GD4 1/20 0.54
VNN1 O95497 4/20 0.53
POLB P06746 1/20 0.53
HSD17B10 Q99714 3/20 0.52
MEN1 O00255 2/20 0.51
LMNA P02545 2/20 0.51
KMT2A Q03164 2/20 0.51
MAPK1 P28482 1/20 0.51
MMP13 P45452 1/20 0.51
HPGD P15428 1/20 0.51
ALDH1A1 P00352 3/20 0.51
SMN1; SMN2 Q16637 1/20 0.50
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31141723 0.89 HDAC3 (0.82) HDAC3HDAC1HDAC2HDAC6PDE5A
SCHEMBL4730176 0.86 HDAC1 (1.00) HDAC3HDAC1HDAC2HDAC6VNN1
SCHEMBL31141597 0.82 ALDH1A1 (0.72) HDAC3HDAC1HDAC2HDAC6PDE5A
SCHEMBL24730682 0.79 VNN1 (0.53) HDAC3HDAC1HDAC2HDAC6PDE5A
SCHEMBL2728973 0.77 AURKA (0.64) HDAC3HDAC1HDAC2HDAC6PDE5A
SCHEMBL7498732 0.76 PDE5A (1.00) PDE5AAURKARPS6KB1AURKBMEN1
SCHEMBL2728976 0.76 AURKA (0.67) HDAC3HDAC1HDAC2HDAC6PDE5A
SCHEMBL7322125 0.75 SMN1; SMN2 (0.68) HSD17B10MEN1LMNAKMT2AMAPK1
SCHEMBL4194265 0.75 AURKA (0.56) HDAC3HDAC1HDAC2HDAC6PDE5A
SCHEMBL13210625 0.72 HPGD (0.69) POLBHSD17B10MEN1LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129802-A1 INHIBITORS OF JAK PORTOLA PHARMACEUTICALS, INC. (US) 2010-11-11 WO claimed