SCHEMBL3797644

SCHEMBL3797644

NC(=O)C1CC(c2nccs2)C1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.37
ALDH1A1 P00352 2/20 0.35
DRD4 P21917 2/20 0.34
KDM4C Q9H3R0 1/20 0.34
GRM5 P41594 1/20 0.34
GRM1 Q13255 1/20 0.34
RBBP9 O75884 1/20 0.34
NOS3 P29474 1/20 0.33
NOS2 P35228 1/20 0.33
MEN1 O00255 1/20 0.33
HTT P42858 1/20 0.33
KMT2A Q03164 1/20 0.33
EPHX2 P34913 1/20 0.33
NPC1 O15118 1/20 0.33
TSHR P16473 1/20 0.33
NOS1 P29475 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GPR88 Q9GZN0 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2053962 0.89 AOC3 (0.37) AOC3ALDH1A1DRD4RBBP9MEN1
SCHEMBL2036893 0.86 RBBP9 (0.39) AOC3ALDH1A1DRD4RBBP9MEN1
SCHEMBL30537972 0.76 HDAC2 (0.36) AOC3ALDH1A1DRD4GRM5GRM1
SCHEMBL2038839 0.76 GPR88 (0.42) AOC3ALDH1A1GRM5GRM1RBBP9
SCHEMBL2014387 0.76 ALDH1A1 (0.34) AOC3ALDH1A1DRD4GRM5GRM1
SCHEMBL2046508 0.75 KDM4E (0.37) AOC3ALDH1A1DRD4KDM4CGRM5
SCHEMBL27842894 0.75 MEN1 (0.43) AOC3ALDH1A1DRD4RBBP9MEN1
SCHEMBL2014210 0.74 KDM4E (0.43) DRD4KDM4CRBBP9MEN1HTT
SCHEMBL2037647 0.74 KDM4E (0.47) DRD4KDM4CRBBP9MEN1HTT
SCHEMBL30343662 0.74 MEN1 (0.36) AOC3DRD4RBBP9MEN1HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010118208-A1 BENZOXAZEPIN-4- (5H) -YL DERIVATIVES AND THEIR USE TO TREAT CANCER EXELIXIS, INC. (US) 2010-10-14 WO disclosed