SCHEMBL3648440

SCHEMBL3648440

CC(C)(C)CN(Cc1cc(-c2cccnc2Cl)c(S(=O)(=O)c2cccnc2)s1)C(=O)O

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GPBAR1 Q8TDU6 1/20 0.38
PTGER2 P43116 9/20 0.35
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
MAPT P10636 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32
SLC40A1 Q9NP59 1/20 0.31
HIF1A Q16665 1/20 0.31
NAMPT P43490 1/20 0.31
KEAP1 Q14145 1/20 0.31
NFE2L2 Q16236 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3650557 0.93 GPBAR1 (0.35) GPBAR1RXFP1SLC40A1NAMPT
SCHEMBL3645990 0.88 PTGER2 (0.35) GPBAR1PTGER2LMNATP53MAPT
SCHEMBL3799201 0.87 PTGER2 (0.35) PTGER2LMNATP53MAPTABCC9
SCHEMBL4130745 0.87 GPBAR1 (0.40) GPBAR1PTGER2LMNATP53MAPT
SCHEMBL3803078 0.83 ALDH1A1 (0.36) LMNAMAPTNAMPT
SCHEMBL3648432 0.82 GPBAR1 (0.39) GPBAR1PTGER2RXFP1ABCC9ABCC8
SCHEMBL3654953 0.81 GPBAR1 (0.33) GPBAR1
SCHEMBL3654310 0.81 GPBAR1 (0.34) GPBAR1PTGER2NAMPT
SCHEMBL3651632 0.80
SCHEMBL3652839 0.80 CTSK (0.32) NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2190822-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS Takeda Pharmaceutical Company Limited (JP) 2010-06-02 EP disclosed
WO-2009041705-A9 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL (JP) 2009-08-13 WO disclosed
WO-2009041705-A2 5-MEMBERED HETEROCYCLIC COMPOUNDS AS PROTON PUMP INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2009-04-02 WO disclosed