SCHEMBL381332

SCHEMBL381332

CNC(=O)ON1CCC(N2CCC(Cc3c(Cl)cc(-c4ccc(C(F)(F)F)cc4)cc3Cl)C2=O)CC1

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.34
CTSS P25774 2/20 0.33
FPR1 P21462 1/20 0.33
FPR2 P25090 1/20 0.33
SCN9A Q15858 1/20 0.32
CNR1 P21554 1/20 0.32
HSD11B1 P28845 1/20 0.31
SLC6A4 P31645 1/20 0.31
HRH3 Q9Y5N1 1/20 0.31
DRD2 P14416 1/20 0.31
DRD4 P21917 1/20 0.31
MGLL Q99685 1/20 0.31
PPARD Q03181 1/20 0.31
PPARA Q07869 1/20 0.31
CHRM3 P20309 1/20 0.31
CCR5 P51681 1/20 0.31
CHRM4 P08173 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL381499 1.00 MCHR1 (0.34) MCHR1CTSSFPR1FPR2SCN9A
SCHEMBL381812 0.91 CHRM3 (0.33) CNR1HSD11B1CHRM3
SCHEMBL381134 0.91 CNR1 (0.36) MCHR1SCN9ACNR1DRD4CHRM3
SCHEMBL380490 0.91 AKR1C2 (0.37) MCHR1SCN9ACHRM3
SCHEMBL381541 0.90 MAPT (0.34) MCHR1HSD11B1HRH3
SCHEMBL381239 0.87 MCHR1 (0.36) MCHR1CTSSFPR1FPR2CNR1
SCHEMBL381008 0.87 MCHR1 (0.36) MCHR1CTSSFPR1FPR2CNR1
SCHEMBL381324 0.86 KIT (0.33)
SCHEMBL380833 0.86 MCHR1 (0.33) MCHR1HSD11B1HRH3CHRM3
SCHEMBL381359 0.86 KIT (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2049513-B1 PIPERIDINYL SUBSTITUTED PYRROLIDINONES AS INHIBITORS OF 11-BETA-HYDROXYSTEROID DEHYDROGENASE 1 LILLY CO ELI (US) 2012-01-25 EP claimed