SCHEMBL3814080

SCHEMBL3814080

O=C(CCCCCc1ccccc1)Nc1ccc2c(c1)COC2=O

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.65
KDM4E B2RXH2 1/20 0.65
ROCK2 O75116 2/20 0.58
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
NFKB1 P19838 1/20 0.57
NFKB2 Q00653 1/20 0.57
RELA Q04206 1/20 0.57
ALDH1A1 P00352 1/20 0.55
RXFP1 Q9HBX9 1/20 0.55
PGR P06401 3/20 0.54
NR3C1 P04150 2/20 0.54
POLB P06746 1/20 0.54
NPSR1 Q6W5P4 1/20 0.54
GAA P10253 1/20 0.53
BRD4 O60885 1/20 0.52
HDAC3 O15379 1/20 0.51
HDAC4 P56524 1/20 0.51
HDAC1 Q13547 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26994672 0.83 MAPT (0.67) MAPTKDM4EROCK2NPC1RAB9A
SCHEMBL6086189 0.76 MAPT (0.71) MAPTKDM4ENPC1SMN1; SMN2ALDH1A1
SCHEMBL28099312 0.76 MAPT (0.74) MAPTKDM4ENPC1RAB9ASMN1; SMN2
SCHEMBL27884806 0.75 KCNJ1 (0.57) MAPTKDM4ERXFP1GAA
SCHEMBL26994676 0.75 MAOA (0.59) MAPTKDM4EALDH1A1RXFP1PGR
SCHEMBL292832 0.75 PGR (0.75) PGRNR3C1NR3C2
SCHEMBL17783820 0.74 ROCK2 (1.00) ROCK2
SCHEMBL29606212 0.73 MAPT (0.66) MAPTKDM4ENPC1ALDH1A1PGR
SCHEMBL4163167 0.73 PGR (0.73) MAPTKDM4EALDH1A1PGRNR3C1
SCHEMBL7831891 0.72 HDAC1 (0.67) MAPTKDM4ENPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2086921-A2 SYNTHESIS OF SELECTED STEREOISOMERS OF CERTAIN SUBSTITUTED ALCOHOLS Bausch & Lomb Incorporated (US) 2009-08-12 EP disclosed
WO-2008060799-A2 SYNTHESIS OF SELECTED STEREOISOMERS OF CERTAIN SUBSTITUTED ALCOHOLS BAUSCH & LOMB INCORPORATED (US) 2008-05-22 WO disclosed