SCHEMBL3815565

SCHEMBL3815565

CC(C)(C)OC(=O)CNc1cccc(CC(c2cccnc2)(c2cccnc2)c2cccc(C#N)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTGER2 P43116 8/20 0.41
GRM5 P41594 4/20 0.38
KCNA5 P22460 2/20 0.36
VNN1 O95497 2/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
ALOX15 P16050 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
CYP2C19 P33261 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CLK4 Q9HAZ1 1/20 0.36
CCNT1 O60563 1/20 0.36
ABCB1 P08183 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1378017 0.83 GRM5 (0.43) GRM5VNN1CYP1A2
SCHEMBL1381950 0.83 CYP1A2 (0.42) PTGER2GRM5VNN1ALDH1A1CYP1A2
SCHEMBL3819011 0.80 HSD11B1 (0.39) PTGER2GRM5KCNA5ALDH1A1CYP1A2
SCHEMBL3818100 0.80 CLK4 (0.36) PTGER2GRM5VNN1ALDH1A1CYP1A2
SCHEMBL1380015 0.75 KCNA5 (0.45) GRM5KCNA5VNN1ALDH1A1CYP1A2
SCHEMBL1378033 0.75 KCNA5 (0.43) PTGER2KCNA5CYP3A4
SCHEMBL1382204 0.73 SMN1; SMN2 (0.42) GRM5ALDH1A1CYP3A4MAPK1
SCHEMBL3813507 0.72 NAMPT (0.42) PTGER2GRM5CYP3A4
SCHEMBL1726534 0.71 ABCB1 (0.45) ALDH1A1CLK4CCNT1ABCB1
SCHEMBL14632483 0.70 ALDH1A1 (0.51) ALDH1A1TSHRMAPK1HSD17B10ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1776355-A4 POTASSIUM CHANNEL INHIBITORS MERCK & CO INC (US) 2009-08-12 EP disclosed
EP-1776355-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2007-04-25 EP disclosed
WO-2006014877-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2006-02-09 WO disclosed